SCHEMBL11352104

SCHEMBL11352104

COC(=O)c1ccc(C(C)CCNCC(O)c2cccc(C(F)(F)F)c2)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB1 P08588 3/20 0.46
ADRB2 P07550 2/20 0.46
ADRB3 P13945 1/20 0.46
KDM4E B2RXH2 1/20 0.44
ALDH1A1 P00352 1/20 0.44
GAA P10253 1/20 0.44
PNMT P11086 1/20 0.43
CCR2 P41597 1/20 0.43
CES2 O00748 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
USP2 O75604 2/20 0.41
CYP3A4 P08684 2/20 0.41
NR1I2 O75469 1/20 0.41
HTR1A P08908 1/20 0.41
ADRA2A P08913 1/20 0.41
ADORA3 P0DMS8 1/20 0.41
ADRA2B P18089 1/20 0.41
ADRA2C P18825 1/20 0.41
CHRM3 P20309 1/20 0.41
SLC6A2 P23975 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11039373 0.85 ADRB1 (0.55) ADRB1ADRB2ADRB3KDM4EGAA
SCHEMBL11043555 0.83 ADRB1 (0.48) ADRB1ADRB2ADRB3KDM4EALDH1A1
SCHEMBL11451326 0.83 ALDH1A1 (0.53) ADRB2ADRB3KDM4EALDH1A1GAA
SCHEMBL11483076 0.83 ALDH1A1 (0.53) ADRB2ADRB3KDM4EALDH1A1GAA
Hydrochloric Acid SCHEMBL11477462 0.82 ALDH1A1 (0.55) ADRB2ADRB3KDM4EALDH1A1GAA
SCHEMBL11039896 0.80 ADRB2 (0.47) ADRB1ADRB2ADRB3KDM4EALDH1A1
SCHEMBL9671378 0.80 POLB (0.49) ADRB1ADRB2ADRB3PNMTCES2
SCHEMBL6540063 0.79 ADRB1 (0.49) ADRB1ADRB2ADRB3KDM4EGAA
SCHEMBL6540069 0.79 ADRB1 (0.49) ADRB1ADRB2ADRB3KDM4EGAA
SCHEMBL9007073 0.78 ADRB3 (0.56) ADRB1ADRB2ADRB3USP2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0021636-A1 Secondary amines, their preparation and use in pharmaceutical compositions BEECHAM GROUP PLC (GB) 1981-01-07 EP disclosed