SCHEMBL11045824

SCHEMBL11045824

CC(=O)SCCC(=O)N1c2ccc(C)cc2CCC1C(=O)ON(C1CCCCC1)C1CCCCC1

nearest known ligand 0.37

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 4/20 0.36
KMT2A Q03164 4/20 0.36
CHRM2 P08172 1/20 0.34
CHRM4 P08173 1/20 0.34
CHRM1 P11229 1/20 0.34
CHRM3 P20309 1/20 0.34
MAPK1 P28482 1/20 0.33
NOTUM Q6P988 1/20 0.33
NPC1 O15118 2/20 0.32
RAB9A P51151 2/20 0.32
ALDH1A1 P00352 1/20 0.32
HTT P42858 1/20 0.32
KDM4E B2RXH2 1/20 0.32
LMNA P02545 1/20 0.32
ACE P12821 1/20 0.32
OPRL1 P41146 1/20 0.31
POLB P06746 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11052123 0.93 MEN1 (0.32) MEN1KMT2ANPC1RAB9ALMNA
SCHEMBL11046009 0.91 MEN1 (0.36) MEN1KMT2AMAPK1NOTUMNPC1
SCHEMBL11051574 0.88 OPRL1 (0.40) CHRM2CHRM4CHRM1CHRM3ACE
SCHEMBL11046064 0.82 ACE (0.42) MAPK1NOTUMACE
SCHEMBL11045822 0.80 MEN1 (0.43) MEN1KMT2ACHRM2CHRM4CHRM1
SCHEMBL11044573 0.78 KMT2A (0.45) KMT2AACEOPRL1
SCHEMBL11050571 0.78 KMT2A (0.45) KMT2AACEOPRL1
SCHEMBL11047878 0.78 KMT2A (0.45) KMT2AACEOPRL1
SCHEMBL11047768 0.76 MTNR1A (0.38) MEN1KMT2AMAPK1NOTUMNPC1
SCHEMBL11043214 0.74 ACE (0.42) KMT2AMAPK1ACE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4461896-A 1-[Acylthio) and (mercapto)-1-oxoalkyl]-1,2,3,4-tetrahydroquinoline-2-carboxylic acids NORWICH EATON PHARMACEUTICALS, INC. (US) 1984-07-24 US disclosed