SCHEMBL11048982

SCHEMBL11048982

COC(=O)Cn1c(=S)[nH]c(=O)c2scc(C)c21

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
QPCT Q16769 3/20 0.35
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
KAT2B Q92831 1/20 0.35
ALDH1A1 P00352 2/20 0.34
HPGD P15428 2/20 0.34
NPSR1 Q6W5P4 2/20 0.34
PPARG P37231 1/20 0.33
NCOA2 Q15596 1/20 0.33
NCOA1 Q15788 1/20 0.33
RXFP1 Q9HBX9 1/20 0.33
NCOA3 Q9Y6Q9 1/20 0.33
HSD17B10 Q99714 1/20 0.33
MAPT P10636 1/20 0.32
MEN1 O00255 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11048979 0.80 QPCT (0.52) KDM4ESMN1; SMN2QPCTNPC1RAB9A
SCHEMBL11045234 0.76 GRIK1 (0.45) KDM4ESMN1; SMN2ALDH1A1HSD17B10MAPT
SCHEMBL11045232 0.68 ALDH1A1 (0.60) SMN1; SMN2QPCTALDH1A1HPGDNPSR1
SCHEMBL23635683 0.64 SMN1; SMN2 (0.44) KDM4ESMN1; SMN2ALDH1A1HPGDNPSR1
SCHEMBL11051146 0.63 SMN1; SMN2 (0.45) KDM4ESMN1; SMN2NPC1RAB9AALDH1A1
SCHEMBL16599416 0.63 MAPK1 (0.38) KDM4EALDH1A1HPGDHSD17B10MAPT
SCHEMBL24961270 0.61 SMN1; SMN2 (0.38) KDM4ESMN1; SMN2NPC1RAB9AALDH1A1
SCHEMBL7643586 0.61 MAPK1 (0.51) HPGDKMT2A
SCHEMBL14198913 0.61 ALDH1A1 (0.41) KDM4ESMN1; SMN2NPC1RAB9AKAT2B
SCHEMBL24703554 0.60 KDM4E (0.57) KDM4ESMN1; SMN2NPC1RAB9AKAT2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4442289-A ANTIASTHMA HOFFMANN-LA ROCHE INC. (US) 1984-04-10 US disclosed
US-4376121-A Antiallerigically-active imidazothienopyrimidine derivatives HOFFMANN-LA ROCHE INC. (US) 1983-03-08 US disclosed