SCHEMBL11053086

SCHEMBL11053086

CNc1ncn(-c2c(C)cc(N)cc2Cl)c(=O)n1

nearest known ligand 0.33

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CHRNA7 P36544 6/20 0.33
PAK1 Q13153 4/20 0.33
EGFR P00533 1/20 0.33
FGFR1 P11362 1/20 0.33
SRC P12931 1/20 0.33
WEE1 P30291 1/20 0.32
PAK2 Q13177 2/20 0.32
SIK2 Q9H0K1 3/20 0.31
SIK1 P57059 2/20 0.31
SIK3 Q9Y2K2 2/20 0.31
STK4 Q13043 1/20 0.30
STK3 Q13188 1/20 0.30
STK26 Q9P289 1/20 0.30
STK24 Q9Y6E0 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11055502 0.91 AURKA (0.32)
SCHEMBL11057711 0.86 EGFR (0.33) PAK1EGFRFGFR1SRCWEE1
SCHEMBL11053102 0.85 HCAR1 (0.34) CHRNA7PAK1EGFRFGFR1SRC
SCHEMBL11053272 0.85 NOS3 (0.32)
SCHEMBL11058843 0.85 MAPK14 (0.31)
SCHEMBL11054473 0.85
SCHEMBL11496851 0.80 SIK1 (0.30) SIK2SIK1SIK3
SCHEMBL11056407 0.79 CRHR1 (0.34) CHRNA7EGFRFGFR1SRC
SCHEMBL11054604 0.79 CHRNA7 (0.47) CHRNA7EGFRFGFR1SRCWEE1
SCHEMBL11058852 0.79 ELANE (0.34)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4452980-A DIARRHEA WILLIAM H. RORER, INC. (US) 1984-06-05 US disclosed
US-4225315-A Triazinones from amidinoureas WILLIAM H. RORER, INC. (US) 1980-09-30 US disclosed