SCHEMBL11060075

SCHEMBL11060075

Cc1cccc(C(F)(F)F)c1-n1cnc(N)nc1=O

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCAR1 Q9BXC0 4/20 0.37
P2RX7 Q99572 2/20 0.37
POLB P06746 2/20 0.36
PARP1 P09874 2/20 0.35
ABL1 P00519 1/20 0.34
LCK P06239 1/20 0.34
KIT P10721 1/20 0.34
SRC P12931 1/20 0.34
PDGFRA P16234 1/20 0.34
HSD11B1 P28845 2/20 0.33
ALDH1A1 P00352 2/20 0.33
C5AR1 P21730 1/20 0.33
XDH P47989 1/20 0.33
MPL P40238 1/20 0.33
AADAT Q8N5Z0 1/20 0.33
KDM4E B2RXH2 1/20 0.33
CYP1A2 P05177 1/20 0.33
HPGD P15428 1/20 0.33
CYP2C19 P33261 1/20 0.33
PIK3CD O00329 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11052581 0.86 HCAR1 (0.48) HCAR1POLBALDH1A1XDH
SCHEMBL11055606 0.86 HCAR1 (0.35) HCAR1P2RX7POLBPARP1XDH
SCHEMBL11054450 0.82 HCAR1 (0.40) HCAR1KDM4E
SCHEMBL11059375 0.82 HCAR1 (0.40) HCAR1XDH
SCHEMBL11055534 0.82 LCK (0.36) HCAR1ABL1LCKKITSRC
SCHEMBL11054591 0.80 CHRNA7 (0.46) HCAR1SRC
SCHEMBL11056476 0.80 HCAR1 (0.40) HCAR1ALDH1A1XDH
SCHEMBL11056242 0.80 HCAR1 (0.40) HCAR1C5AR1
SCHEMBL11056827 0.80 HCAR1 (0.36) HCAR1ABL1LCKKITSRC
SCHEMBL11057681 0.77 APLNR (0.39) HCAR1POLBALDH1A1KDM4EHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4452980-A DIARRHEA WILLIAM H. RORER, INC. (US) 1984-06-05 US disclosed
US-4246409-A ANTIDIARRHEAL AGENTS WILLIAM H. RORER, INC. (US) 1981-01-20 US disclosed