SCHEMBL11059375

SCHEMBL11059375

Cc1cccc(I)c1-n1cnc(N)nc1=O

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HCAR1 Q9BXC0 5/20 0.40
DPP4 P27487 2/20 0.33
ANPEP P15144 1/20 0.33
KMT2A Q03164 1/20 0.32
ROCK1 Q13464 1/20 0.32
CHRNA7 P36544 4/20 0.32
PDGFRB P09619 1/20 0.32
XDH P47989 1/20 0.32
C1R P00736 1/20 0.32
FGFR1 P11362 1/20 0.31
CLK1 P49759 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11052581 0.90 HCAR1 (0.48) HCAR1DPP4ANPEPKMT2ACHRNA7
SCHEMBL11054450 0.83 HCAR1 (0.40) HCAR1DPP4CHRNA7
SCHEMBL11056476 0.83 HCAR1 (0.40) HCAR1DPP4ANPEPKMT2ACHRNA7
SCHEMBL11056242 0.83 HCAR1 (0.40) HCAR1DPP4ANPEPKMT2ACHRNA7
SCHEMBL11054591 0.83 CHRNA7 (0.46) HCAR1KMT2ACHRNA7FGFR1
SCHEMBL11060075 0.82 HCAR1 (0.37) HCAR1XDH
SCHEMBL11057681 0.81 APLNR (0.39) HCAR1KMT2AFGFR1
SCHEMBL11057576 0.81 ALDH1A1 (0.39) HCAR1DPP4ANPEP
SCHEMBL11050203 0.80 HCAR1 (0.37) HCAR1CHRNA7
SCHEMBL11055224 0.80 HCAR1 (0.37) HCAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4452980-A DIARRHEA WILLIAM H. RORER, INC. (US) 1984-06-05 US disclosed
US-4246409-A ANTIDIARRHEAL AGENTS WILLIAM H. RORER, INC. (US) 1981-01-20 US disclosed
US-4225315-A Triazinones from amidinoureas WILLIAM H. RORER, INC. (US) 1980-09-30 US disclosed