SCHEMBL11056476

SCHEMBL11056476

Cc1cccc(Br)c1-n1cnc(N)nc1=O

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HCAR1 Q9BXC0 4/20 0.40
DPP4 P27487 2/20 0.33
WEE1 P30291 1/20 0.33
ANPEP P15144 1/20 0.33
KMT2A Q03164 1/20 0.32
CHRNA7 P36544 4/20 0.32
ALDH1A1 P00352 1/20 0.32
PDE7A Q13946 1/20 0.32
XDH P47989 1/20 0.32
FGFR1 P11362 1/20 0.31
PKMYT1 Q99640 2/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2D6 P10635 1/20 0.31
CYP2C9 P11712 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11052581 0.90 HCAR1 (0.48) HCAR1DPP4ANPEPKMT2ACHRNA7
SCHEMBL11055375 0.84 GABRA1 (0.36) HCAR1DPP4ANPEPALDH1A1FGFR1
SCHEMBL11054591 0.83 CHRNA7 (0.46) HCAR1KMT2ACHRNA7FGFR1
SCHEMBL11059375 0.83 HCAR1 (0.40) HCAR1DPP4ANPEPKMT2ACHRNA7
SCHEMBL11056242 0.83 HCAR1 (0.40) HCAR1DPP4ANPEPKMT2ACHRNA7
SCHEMBL11054450 0.83 HCAR1 (0.40) HCAR1DPP4CHRNA7PDE7A
SCHEMBL11053171 0.81 ELANE (0.33) HCAR1ALDH1A1
SCHEMBL11057681 0.81 APLNR (0.39) HCAR1KMT2AALDH1A1FGFR1
SCHEMBL11053236 0.81 HCAR1 (0.38) HCAR1WEE1KMT2ACHRNA7ALDH1A1
SCHEMBL11057576 0.81 ALDH1A1 (0.39) HCAR1DPP4ANPEPALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4452980-A DIARRHEA WILLIAM H. RORER, INC. (US) 1984-06-05 US disclosed
US-4246409-A ANTIDIARRHEAL AGENTS WILLIAM H. RORER, INC. (US) 1981-01-20 US disclosed
US-4225315-A Triazinones from amidinoureas WILLIAM H. RORER, INC. (US) 1980-09-30 US disclosed