SCHEMBL11060167

SCHEMBL11060167

CCc1cccc(Cl)c1-n1cnc(N(CC)CC)nc1=O

nearest known ligand 0.38

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.38
HCAR1 Q9BXC0 2/20 0.37
POLB P06746 1/20 0.37
MAPK14 Q16539 2/20 0.35
CHRNA7 P36544 6/20 0.35
MAPK11 Q15759 1/20 0.34
SMN1; SMN2 Q16637 4/20 0.33
LMNA P02545 1/20 0.33
ALDH1A1 P00352 1/20 0.33
ALOX15 P16050 1/20 0.33
TSHR P16473 1/20 0.32
HTT P42858 1/20 0.32
RXFP1 Q9HBX9 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11058424 0.90 HCAR1 (0.37) TDP1HCAR1SMN1; SMN2LMNAALDH1A1
SCHEMBL11050218 0.90 HCAR1 (0.37) HCAR1POLBMAPK14CHRNA7MAPK11
SCHEMBL11055569 0.88 CHRNA7 (0.43) TDP1HCAR1CHRNA7
SCHEMBL11055471 0.85 HCAR1 (0.38) HCAR1CHRNA7SMN1; SMN2ALOX15
SCHEMBL11055617 0.81 FGFR1 (0.39) HCAR1MAPK14CHRNA7MAPK11
SCHEMBL11347343 0.81 ANPEP (0.36) HCAR1LMNAALDH1A1
SCHEMBL11053513 0.80 MAPK14 (0.39) MAPK14CHRNA7ALDH1A1
SCHEMBL11056331 0.79 MAT2A (0.41) HCAR1LMNAALDH1A1TSHR
SCHEMBL11359839 0.79 SLC29A1 (0.36) HCAR1LMNAALDH1A1HTT
SCHEMBL11058764 0.79 FGFR1 (0.41) HCAR1MAPK14CHRNA7MAPK11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4452980-A DIARRHEA WILLIAM H. RORER, INC. (US) 1984-06-05 US disclosed
US-4246409-A ANTIDIARRHEAL AGENTS WILLIAM H. RORER, INC. (US) 1981-01-20 US disclosed
US-4225315-A Triazinones from amidinoureas WILLIAM H. RORER, INC. (US) 1980-09-30 US disclosed