SCHEMBL11060209

SCHEMBL11060209

CCCN(CCC)c1ncn(-c2c(C)cccc2C)c(=O)n1

nearest known ligand 0.41

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HCAR1 Q9BXC0 1/20 0.41
CRHR1 P34998 14/20 0.38
ELANE P08246 1/20 0.34
MAPT P10636 1/20 0.33
ALOX15 P16050 1/20 0.32
CREBBP Q92793 1/20 0.32
TP53 P04637 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11056383 0.96 HCAR1 (0.40) HCAR1CRHR1ELANEALOX15CREBBP
SCHEMBL11052461 0.88 HCAR1 (0.40) HCAR1CRHR1ELANETP53
SCHEMBL11059494 0.84 CRHR1 (0.38) HCAR1CRHR1
SCHEMBL11055471 0.84 HCAR1 (0.38) HCAR1CRHR1ELANEALOX15TP53
SCHEMBL11059656 0.83 HCAR1 (0.43) HCAR1
SCHEMBL11401770 0.83 HCAR1 (0.39) HCAR1CRHR1ELANEMAPTTP53
SCHEMBL11059289 0.82 HCAR1 (0.36) HCAR1CRHR1ALOX15
SCHEMBL11053245 0.82 CHRNA7 (0.41) HCAR1CRHR1MAPTTP53
SCHEMBL11055569 0.82 CHRNA7 (0.43) HCAR1
SCHEMBL11056926 0.81 HCAR1 (0.46) HCAR1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4452980-A DIARRHEA WILLIAM H. RORER, INC. (US) 1984-06-05 US disclosed
US-4246409-A ANTIDIARRHEAL AGENTS WILLIAM H. RORER, INC. (US) 1981-01-20 US disclosed
US-4225315-A Triazinones from amidinoureas WILLIAM H. RORER, INC. (US) 1980-09-30 US disclosed