SCHEMBL11059289

SCHEMBL11059289

CCN(CC)c1ncn(-c2c(C)cccc2Br)c(=O)n1

nearest known ligand 0.36

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HCAR1 Q9BXC0 3/20 0.36
ALOX15 P16050 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
GRIN1 Q05586 2/20 0.31
GRIN2A Q12879 2/20 0.31
GBA1 P04062 1/20 0.31
HTR2C P28335 2/20 0.31
HTR2A P28223 1/20 0.31
CRHR1 P34998 3/20 0.31
CHRNA7 P36544 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11055971 0.89 HCAR1 (0.36) HCAR1CHRNA7
SCHEMBL11055471 0.87 HCAR1 (0.38) HCAR1ALOX15SMN1; SMN2GRIN1GRIN2A
SCHEMBL11053236 0.87 HCAR1 (0.38) HCAR1CHRNA7
SCHEMBL11055569 0.85 CHRNA7 (0.43) HCAR1CHRNA7
SCHEMBL11056383 0.83 HCAR1 (0.40) HCAR1ALOX15CRHR1
SCHEMBL11060209 0.82 HCAR1 (0.41) HCAR1ALOX15CRHR1
SCHEMBL11058424 0.81 HCAR1 (0.37) HCAR1ALOX15SMN1; SMN2GRIN1GRIN2A
SCHEMBL11057683 0.80 MAPK14 (0.34) HCAR1SMN1; SMN2CHRNA7
SCHEMBL11056476 0.79 HCAR1 (0.40) HCAR1CHRNA7
SCHEMBL11059656 0.79 HCAR1 (0.43) HCAR1SMN1; SMN2CHRNA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4452980-A DIARRHEA WILLIAM H. RORER, INC. (US) 1984-06-05 US disclosed
US-4246409-A ANTIDIARRHEAL AGENTS WILLIAM H. RORER, INC. (US) 1981-01-20 US disclosed
US-4225315-A Triazinones from amidinoureas WILLIAM H. RORER, INC. (US) 1980-09-30 US disclosed