SCHEMBL11060675

SCHEMBL11060675

CCCCOc1ncncc1N(S)C(N)=O

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.33
KMT2A Q03164 2/20 0.33
CYP3A4 P08684 2/20 0.33
CA12 O43570 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA9 Q16790 1/20 0.33
MEN1 O00255 1/20 0.33
NR1I2 O75469 1/20 0.33
CHRM2 P08172 1/20 0.33
ADRA2A P08913 1/20 0.33
MAPT P10636 1/20 0.33
OPRK1 P41145 1/20 0.33
HTR2B P41595 1/20 0.33
SLC6A3 Q01959 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
TSHR P16473 2/20 0.33
L3MBTL1 Q9Y468 2/20 0.33
CYP1A2 P05177 2/20 0.33
CYP2C9 P11712 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11058190 0.87 PARP10 (0.32) TSHRMKNK2
SCHEMBL11058669 0.81 GPBAR1 (0.33) CDC7CDK2
SCHEMBL11062439 0.81 GABRP (0.35) LMNAKMT2ACYP3A4MEN1MAPT
SCHEMBL11061057 0.80 MAP3K7 (0.37) LMNAKMT2ACYP3A4CA12CA1
SCHEMBL11058625 0.78 MAP3K7 (0.36) MAP3K7TAB1GSK3B
SCHEMBL11055926 0.76 SMN1; SMN2 (0.35) LMNAKMT2ACYP3A4CA12CA1
SCHEMBL11060945 0.76 RPS6KB1 (0.30) RPS6KB1
SCHEMBL11058684 0.75 LMNA (0.43) LMNAKMT2ACYP3A4MEN1NR1I2
SCHEMBL11060720 0.74 CYP3A4 (0.36) LMNAKMT2ACYP3A4MEN1NR1I2
SCHEMBL11058664 0.73

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4434167-A Pyrimidyl thioureas useful for the treatment of hypertension and hyperlipidemia BEIERSDORF AKTIENGESELLSCHAFT (DE) 1984-02-28 US disclosed