SCHEMBL11060720

SCHEMBL11060720

CCCCCOc1nc(OC)ncc1N(S)C(N)=O

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.36
MEN1 O00255 1/20 0.36
NR1I2 O75469 1/20 0.36
LMNA P02545 1/20 0.36
CHRM2 P08172 1/20 0.36
ADRA2A P08913 1/20 0.36
MAPT P10636 1/20 0.36
OPRK1 P41145 1/20 0.36
HTR2B P41595 1/20 0.36
SLC6A3 Q01959 1/20 0.36
KMT2A Q03164 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
PLAU P00749 1/20 0.33
ACACB O00763 1/20 0.33
SMPD1 P17405 3/20 0.32
GABRG2 P18507 1/20 0.32
GABRB3 P28472 1/20 0.32
GABRA2 P47869 1/20 0.32
CDK1 P06493 1/20 0.32
CCNB1 P14635 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10959345 0.84 PLAU (0.41) PLAUACACBGABRG2GABRB3GABRA2
SCHEMBL11061481 0.80 PLAU (0.33) MEN1KMT2APLAUACACBGABRG2
SCHEMBL11061001 0.79 MEN1 (0.35) MEN1KMT2AACACB
SCHEMBL11064906 0.77 MAP3K7 (0.32) MEN1LMNAMAPTKMT2ACDK1
SCHEMBL11060675 0.74 LMNA (0.33) CYP3A4MEN1NR1I2LMNACHRM2
SCHEMBL11063674 0.73 CYP3A4 (0.38) CYP3A4MEN1NR1I2LMNACHRM2
SCHEMBL11058684 0.71 LMNA (0.43) CYP3A4MEN1NR1I2LMNACHRM2
SCHEMBL11059949 0.71 ACACB (0.33) ACACB
SCHEMBL11060716 0.70 MEN1 (0.36) CYP3A4MEN1NR1I2LMNACHRM2
SCHEMBL11055926 0.69 SMN1; SMN2 (0.35) CYP3A4MEN1NR1I2LMNACHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4434167-A Pyrimidyl thioureas useful for the treatment of hypertension and hyperlipidemia BEIERSDORF AKTIENGESELLSCHAFT (DE) 1984-02-28 US disclosed