SCHEMBL11064972

SCHEMBL11064972

CC(C)C(N)C(=O)OCc1cccc(C(=O)c2ccccc2)n1

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.39
CNR2 P34972 1/20 0.38
MRGPRX4 Q96LA9 3/20 0.37
KMT2A Q03164 1/20 0.37
SLC15A1 P46059 1/20 0.37
GLS O94925 1/20 0.36
ELANE P08246 1/20 0.36
PTGS1 P23219 1/20 0.36
PTGS2 P35354 1/20 0.36
PDE5A O76074 3/20 0.36
PDE1A P54750 1/20 0.36
PDE1B Q01064 1/20 0.36
PDE1C Q14123 1/20 0.36
ALDH1A1 P00352 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11462428 0.82 ALOX5 (0.39) CNR2MRGPRX4PTGS1PTGS2PDE5A
SCHEMBL11472173 0.81 ALDH1A1 (0.47) BRD4CNR2MRGPRX4KMT2AELANE
SCHEMBL11064786 0.79 POLB (0.36) BRD4MRGPRX4KMT2APTGS1PTGS2
SCHEMBL11062094 0.78 KCNH2 (0.38) SLC15A1PTGS1ALDH1A1
SCHEMBL11471667 0.77 MRGPRX4 (0.43) BRD4CNR2MRGPRX4KMT2APTGS2
SCHEMBL11069825 0.75 PDE5A (0.36) BRD4MRGPRX4KMT2APDE5APDE1A
SCHEMBL11069822 0.75 PDE5A (0.36) BRD4MRGPRX4KMT2APDE5APDE1A
SCHEMBL11392950 0.75 NOS3 (0.35) BRD4CNR2KMT2APDE5APDE1A
SCHEMBL11392948 0.75 NOS3 (0.35) BRD4CNR2KMT2APDE5APDE1A
SCHEMBL11403555 0.75 MRGPRX4 (0.42) CNR2MRGPRX4PDE5APDE1APDE1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4447613-A Pyridyl esters and thiolesters of aminoalkanoic acids ZOECON CORPORATION (US) 1984-05-08 US disclosed
US-4269981-A Certain pyridylmethyl esters of formamido-lower-alkanoates and derivatives thereof ZOECON CORPORATION (US) 1981-05-26 US disclosed
US-4247701-A Certain pesticidal substituted amino lower-alkanoates or lower-alkano-thioates containing pyridyl in the ester portion ZOECON CORPORATION (US) 1981-01-27 US disclosed