SCHEMBL11069932

SCHEMBL11069932

Cc1ccc(C2(N(C)C)CCC(=O)C(C)C2)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRL1 P41146 8/20 0.41
OPRM1 P35372 7/20 0.41
OPRK1 P41145 2/20 0.41
MAOB P27338 4/20 0.39
MAOA P21397 2/20 0.39
SLC6A2 P23975 2/20 0.34
SLC6A3 Q01959 2/20 0.34
SLC6A4 P31645 1/20 0.34
KCNH2 Q12809 1/20 0.34
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
CCR2 P41597 1/20 0.33
CHRNA1 P02708 1/20 0.32
CHRNG P07510 1/20 0.32
CHRNB1 P11230 1/20 0.32
CHRNB2 P17787 1/20 0.32
CHRNB4 P30926 1/20 0.32
CHRNA3 P32297 1/20 0.32
CHRNA4 P43681 1/20 0.32
CHRND Q07001 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11090331 0.86 MAOA (0.38) OPRL1OPRM1OPRK1MAOBMAOA
SCHEMBL11070605 0.86 MAOA (0.38) OPRL1OPRM1OPRK1MAOBMAOA
SCHEMBL11096526 0.86 MAOA (0.38) OPRL1OPRM1OPRK1MAOBMAOA
SCHEMBL2440151 0.86 OPRL1 (0.52) OPRL1OPRM1OPRK1
SCHEMBL11090323 0.81 OPRM1 (0.38) OPRL1OPRM1OPRK1MAOBMAOA
SCHEMBL11078629 0.76 OPRL1 (0.51) OPRL1OPRM1OPRK1MAOBMAOA
SCHEMBL11097552 0.76 OPRK1 (0.41) OPRM1OPRK1SLC6A2SLC6A4MEN1
SCHEMBL11078172 0.75 MAOA (0.33) MAOBMAOASLC6A2SLC6A3SLC6A4
SCHEMBL11069388 0.73 SLC6A4 (0.33) OPRL1OPRM1MAOBMAOASLC6A2
SCHEMBL3407450 0.72 OPRL1 (0.54) OPRL1OPRM1OPRK1MAOBMAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4460604-A ANALGESICS, NARCOTIC ANTAGONIST THE UPJOHN COMPANY (US) 1984-07-17 US disclosed
US-4447454-A Analgetic compounds, compositions and process of treatment THE UPJOHN COMPANY (US) 1984-05-08 US disclosed
US-4180584-A ANALGESIC; NARCOTIC ANTAGONIST THE UPJOHN COMPANY (US) 1979-12-25 US disclosed
US-4113866-A ANALGETIC COMPOUNDS, COMPOSITIONS AND PROCESS OF TREATMENT THE UPJOHN COMPANY (US) 1978-09-12 US disclosed
US-4065573-A ANALGESICS THE UPJOHN COMPANY (US) 1977-12-27 US disclosed