SCHEMBL11071000

SCHEMBL11071000

CC(C(=O)NC1CCCCC1)N1CCNCC1

nearest known ligand 0.65

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.65
SIGMAR1 Q99720 4/20 0.63
ALDH1A1 P00352 1/20 0.52
CHRM5 P08912 1/20 0.51
CHRM3 P20309 1/20 0.51
EPHX1 P07099 2/20 0.49
HTT P42858 2/20 0.47
GAA P10253 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
EPHX2 P34913 2/20 0.44
TSHR P16473 2/20 0.44
ATM Q13315 1/20 0.43
LMNA P02545 1/20 0.43
CASP6 P55212 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL977989 0.95 KDM4E (0.58) KDM4ESIGMAR1ALDH1A1CHRM5CHRM3
SCHEMBL1021506 0.94 KDM4E (0.58) KDM4ESIGMAR1ALDH1A1CHRM5CHRM3
SCHEMBL1899938 0.92 KDM4E (0.54) KDM4ESIGMAR1ALDH1A1CHRM5CHRM3
SCHEMBL983313 0.81 SIGMAR1 (0.78) KDM4ESIGMAR1CHRM5CHRM3EPHX1
SCHEMBL24322648 0.78 SIGMAR1 (0.76) KDM4ESIGMAR1ALDH1A1EPHX1GAA
SCHEMBL974058 0.77 SIGMAR1 (1.00) KDM4ESIGMAR1CHRM5CHRM3EPHX1
SCHEMBL29955444 0.77 KDM4E (0.59) KDM4ESIGMAR1ALDH1A1EPHX1HTT
SCHEMBL11063231 0.76 SIGMAR1 (0.54) KDM4ESIGMAR1ALDH1A1CHRM5CHRM3
SCHEMBL973523 0.76 SIGMAR1 (1.00) KDM4ESIGMAR1ALDH1A1CHRM5CHRM3
Hydrochloric Acid SCHEMBL5485542 0.75 SIGMAR1 (0.52) KDM4ESIGMAR1ALDH1A1CHRM5CHRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4478838-A VASODILATOR AGENTS HOKURIKU PHARMACEUTICAL CO., LTD. (JP) 1984-10-23 US disclosed
EP-0083712-A1 1-(3,4,5-Trimethoxycinnamoyl)-4-aminocarbonylethyl-substituted piperazine derivatives and a process for the preparation thereof Hokuriku Pharmaceutical Co.,Ltd (JP) 1983-07-20 EP disclosed