SCHEMBL974058

SCHEMBL974058

CCCCC(C(=O)NC1CCCCC1)N1CCNCC1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 4/20 1.00
CHRM5 P08912 1/20 0.48
CHRM3 P20309 1/20 0.48
KDM4E B2RXH2 2/20 0.44
EPHX1 P07099 10/20 0.43
EPHX2 P34913 2/20 0.42
GNAI3 P08754 1/20 0.41
GNAO1 P09471 1/20 0.41
GNAI1 P63096 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL983313 0.88 SIGMAR1 (0.78) SIGMAR1CHRM5CHRM3KDM4EEPHX1
SCHEMBL11071000 0.77 KDM4E (0.65) SIGMAR1CHRM5CHRM3KDM4EEPHX1
SCHEMBL28816385 0.75 SIGMAR1 (0.59) SIGMAR1GNAI3GNAO1GNAI1
SCHEMBL6324945 0.74 SIGMAR1 (0.58) SIGMAR1KDM4EEPHX1EPHX2
SCHEMBL1900357 0.74 SIGMAR1 (0.58) SIGMAR1CHRM5CHRM3GNAI3GNAO1
SCHEMBL9825772 0.73 SIGMAR1 (0.57) SIGMAR1KDM4EEPHX1EPHX2
SCHEMBL977989 0.73 KDM4E (0.58) SIGMAR1CHRM5CHRM3KDM4EEPHX1
SCHEMBL10103544 0.73 SIGMAR1 (0.57) SIGMAR1KDM4EEPHX1EPHX2
SCHEMBL1021506 0.72 KDM4E (0.58) SIGMAR1CHRM5CHRM3KDM4EEPHX1
SCHEMBL11354516 0.71 SIGMAR1 (0.55) SIGMAR1EPHX1EPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011000945-A9 AMINOALKAMIDES FOR USE IN THE TREATMENT OF INFLAMMATORY, DEGENERATIVE OR DEMYELINATING DISEASES OF THE CNS NENSIUS RESEARCH A/S (DK) 2011-04-07 WO claimed
WO-2011000945-A9 AMINOALKAMIDES FOR USE IN THE TREATMENT OF INFLAMMATORY, DEGENERATIVE OR DEMYELINATING DISEASES OF THE CNS NENSIUS RESEARCH A/S (DK) 2011-04-07 WO disclosed
WO-2011000945-A2 AMINOALKAMIDES FOR USE IN THE TREATMENT OF INFLAMMATORY, DEGENERATIVE OR DEMYELINATING DISEASES OF THE CNS NENSIUS RESEARCH A/S (DK) 2011-01-06 WO disclosed