SCHEMBL11074405

SCHEMBL11074405

CN1CCC(c2ccc(N(C)C)cc2)(C(C)(C)O)CC1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRL1 P41146 1/20 0.39
SLC2A1 P11166 1/20 0.38
CCR1 P32246 1/20 0.36
DRD2 P14416 1/20 0.34
HSD17B10 Q99714 5/20 0.34
ALDH1A1 P00352 4/20 0.34
TSHR P16473 2/20 0.34
ALOX15 P16050 1/20 0.34
CYP3A4 P08684 3/20 0.33
CYP1A2 P05177 3/20 0.33
KDM4E B2RXH2 2/20 0.33
MAPT P10636 2/20 0.33
HPGD P15428 2/20 0.33
CYP2D6 P10635 2/20 0.33
MAPK1 P28482 2/20 0.33
TP53 P04637 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
GLA P06280 1/20 0.33
USP2 O75604 1/20 0.33
CASP1 P29466 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10640876 0.82 OPRM1 (0.49) OPRL1CYP1A2OPRM1OPRD1
SCHEMBL10637592 0.81 OPRM1 (0.46) DRD2ALDH1A1KDM4EMAPTCYP2D6
SCHEMBL10637222 0.81 OPRM1 (0.50) DRD2ALDH1A1MAPTOPRM1
SCHEMBL1152677 0.80 OPRM1 (0.49) DRD2ALDH1A1TSHRMAPTOPRM1
SCHEMBL11068281 0.78 ALDH1A1 (0.43) CCR1DRD2HSD17B10ALDH1A1TSHR
SCHEMBL10641018 0.78 POLB (0.42) TSHRMAPTMAPK1SMN1; SMN2OPRM1
SCHEMBL11074351 0.78 SLC6A4 (0.43) OPRL1CYP3A4MAPTCYP2C19OPRM1
SCHEMBL11073037 0.75 MMP2 (0.46) MAPTSMN1; SMN2HRH4OPRM1OPRD1
SCHEMBL5754493 0.72 CHRM1 (0.37) DRD2HRH4OPRM1OPRD1
SCHEMBL11075430 0.71 OPRD1 (0.44) OPRL1OPRM1OPRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4485109-A 4-Aryl-4-piperidinecarbinols E. I. DU PONT DE NEMOURS AND COMPANY (US) 1984-11-27 US disclosed
EP-0094018-A2 4-Aryl-4-piperidinecarbinols E.I. DU PONT DE NEMOURS AND COMPANY (US) 1983-11-16 EP disclosed