SCHEMBL11082017

SCHEMBL11082017

CC(C)(C)OC(=O)N1CCN(CC(=O)O)C(=O)C1Cc1ccc(OCc2ccccc2)cc1

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
YAP1 P46937 3/20 0.47
LMNA P02545 1/20 0.45
ITGB3 P05106 1/20 0.45
ITGA2B P08514 1/20 0.45
GHSR Q92847 5/20 0.44
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
KDM4C Q9H3R0 1/20 0.43
PLA2G10 O15496 1/20 0.43
PLA2G5 P39877 1/20 0.43
NR1H2 P55055 2/20 0.41
NR1H3 Q13133 2/20 0.41
MCL1 Q07820 1/20 0.41
GPR119 Q8TDV5 2/20 0.41
PARP1 P09874 1/20 0.41
PRMT5 O14744 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11080546 0.92 YAP1 (0.49) YAP1LMNAITGB3ITGA2BGHSR
SCHEMBL11084132 0.91 ITGB3 (0.52) ITGB3ITGA2BKMT2APLA2G10PLA2G5
SCHEMBL11084218 0.84 ITGB3 (0.43) ITGB3ITGA2BMEN1KMT2APLA2G10
SCHEMBL11077466 0.82 PLA2G10 (0.52) ITGB3ITGA2BPLA2G10PLA2G5NR1H2
SCHEMBL11078135 0.81 LMNA (0.47) YAP1LMNAGHSRMEN1KMT2A
SCHEMBL6936067 0.77 PLA2G10 (0.54) MEN1KMT2APLA2G10PLA2G5NR1H2
SCHEMBL7650079 0.76 PLA2G10 (0.41) ITGB3ITGA2BMEN1KMT2APLA2G10
SCHEMBL5043388 0.75 ABHD6 (0.43) YAP1GHSRPLA2G10PLA2G5NR1H2
SCHEMBL11088457 0.75 HTT (0.40) YAP1ITGB3ITGA2BGHSRMEN1
SCHEMBL11078872 0.75 CCR3 (0.44) ITGB3ITGA2BMEN1KMT2APLA2G10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4483988-A Substituted derivatives of 4-t-alkoxycarbonyl-piperazin-2-ones RICHARDSON MERRELL INC. (US) 1984-11-20 US disclosed
US-4435571-A 5-(Substituted benzyl)-6-oxo-2-piperazine carboxylic acids and esters RICHARDSON MERRELL INC. (US) 1984-03-06 US disclosed
US-4341698-A Enkaphalin derivatives RICHARDSON-MERRELL INC. (US) 1982-07-27 US disclosed