SCHEMBL11088975

SCHEMBL11088975

CCOC(=O)c1cn2c(nc1=O)CCC2

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 3/20 0.57
HSD17B10 Q99714 3/20 0.57
TP53 P04637 3/20 0.57
KDM4E B2RXH2 5/20 0.44
MAPT P10636 4/20 0.44
POLB P06746 2/20 0.43
ALDH1A1 P00352 4/20 0.42
GAA P10253 3/20 0.42
NPC1 O15118 2/20 0.42
RAB9A P51151 2/20 0.42
GLA P06280 2/20 0.42
CYP1A2 P05177 1/20 0.42
CYP2C19 P33261 1/20 0.42
L3MBTL1 Q9Y468 2/20 0.41
P2RX7 Q99572 1/20 0.41
KMT2A Q03164 3/20 0.41
MEN1 O00255 2/20 0.41
LMNA P02545 3/20 0.40
PDE3B Q13370 1/20 0.40
PDE3A Q14432 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11182694 0.95 HSD17B10 (0.52) HPGDHSD17B10TP53KDM4EMAPT
SCHEMBL12443590 0.83 HPGD (0.60) HPGDHSD17B10TP53KDM4EMAPT
SCHEMBL13424113 0.79 HPGD (0.55) HPGDHSD17B10TP53KDM4EMAPT
SCHEMBL11097275 0.77 WDR5 (0.46) HPGDHSD17B10TP53KDM4EMAPT
SCHEMBL11089313 0.76 WDR5 (0.42) HPGDHSD17B10TP53KDM4EMAPT
SCHEMBL11089476 0.76 ALDH1A1 (0.40) HPGDHSD17B10TP53KDM4EMAPT
SCHEMBL11093896 0.75 WDR5 (0.42) HPGDHSD17B10TP53KDM4EMAPT
SCHEMBL31355725 0.75 ALDH1A1 (0.42) HPGDHSD17B10TP53KDM4EMAPT
Iodide SCHEMBL11088676 0.75 AKR1C3 (0.41) HPGDHSD17B10TP53KDM4EMAPT
SCHEMBL11087009 0.73 WDR5 (0.47) HPGDHSD17B10TP53KDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4482557-A 3-Substituted-2-oxo-tetrahydro-pyrrol[1,2-a]pyrimidines having digitalis-like activity CHINOIN GYOGYSZER ES VEGYESZETI TERMEKEK GYARA RT. (HU) 1984-11-13 US claimed
US-4482557-A 3-Substituted-2-oxo-tetrahydro-pyrrol[1,2-a]pyrimidines having digitalis-like activity CHINOIN GYOGYSZER ES VEGYESZETI TERMEKEK GYARA RT. (HU) 1984-11-13 US disclosed
US-4367229-A 3-Substituted-tetrahydro-pyrrolo[1,2-a]pyrimidines and pharmaceutical compositions CHINOIN GYOGYSZER ES VEGYESZETI TERMEKEK GYARA RT. (HU) 1983-01-04 US disclosed