SCHEMBL11095481

SCHEMBL11095481

NC(=O)c1cc2c(ccc3cccnc32)[nH]c1=O

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 6/20 0.54
KDM4E B2RXH2 2/20 0.43
TET2 Q6N021 1/20 0.42
TET1 Q8NFU7 1/20 0.42
PLK4 O00444 1/20 0.42
MAP4K4 O95819 1/20 0.42
EGFR P00533 1/20 0.42
ROS1 P08922 1/20 0.42
PIM1 P11309 1/20 0.42
AXL P30530 1/20 0.42
FLT3 P36888 1/20 0.42
FRK P42685 1/20 0.42
MAP4K2 Q12851 1/20 0.42
NTRK3 Q16288 1/20 0.42
MINK1 Q8N4C8 1/20 0.42
AURKB Q96GD4 1/20 0.42
HIPK2 Q9H2X6 1/20 0.42
MKNK2 Q9HBH9 1/20 0.42
IRAK4 Q9NWZ3 1/20 0.42
STK17A Q9UEE5 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7345653 0.89 PARP1 (0.46) PARP1KDM4ETET2TET1ALDH1A1
SCHEMBL7345844 0.80 ALDH1A1 (0.55) PARP1KDM4EPIM1ALDH1A1LMNA
SCHEMBL7348155 0.76 DAO (0.44) PARP1KDM4EHTTTDP1DAO
SCHEMBL16463537 0.76 DAO (0.62) PARP1KDM4EMAPTTDP1JAK2
SCHEMBL1210670 0.76 DAO (0.62) PARP1MAPTSMN1; SMN2RIPK1DAO
SCHEMBL10964234 0.75 CSNK2A1 (0.41) PARP1KDM4EJAK2DAO
SCHEMBL7339417 0.74 PARP1 (0.47) PARP1KDM4EALDH1A1SLC40A1LMNA
SCHEMBL10811949 0.73 KDM4E (0.56) PARP1KDM4EALDH1A1TSHRHTT
SCHEMBL7341890 0.72 PARP1 (0.44) PARP1KDM4ELMNAHSP90AA1CYP3A4
SCHEMBL7337387 0.71 ALDH1A1 (0.51) PARP1KDM4EALDH1A1LMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0102046-A1 Tricyclic lactams, method for making them, pharmaceutical compositions containing them SCHERING CORPORATION (US) 1984-03-07 EP disclosed