SCHEMBL7337387

SCHEMBL7337387

N=C(N)c1cc2c(ccc3ccccc32)[nH]c1=O

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.51
KDM4E B2RXH2 4/20 0.51
LMNA P02545 2/20 0.51
HSD17B10 Q99714 2/20 0.51
PARP1 P09874 7/20 0.46
GRIN2D O15399 1/20 0.41
GRIN3B O60391 1/20 0.41
GRIN1 Q05586 1/20 0.41
GRIN2A Q12879 1/20 0.41
GRIN2B Q13224 1/20 0.41
GRIN2C Q14957 1/20 0.41
GRIN3A Q8TCU5 1/20 0.41
MAPT P10636 2/20 0.40
IDE P14735 1/20 0.40
MPI P34949 1/20 0.40
CACNA1B Q00975 1/20 0.40
APBA1 Q02410 1/20 0.40
BRD4 O60885 3/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7345844 0.88 ALDH1A1 (0.55) ALDH1A1KDM4ELMNAHSD17B10PARP1
SCHEMBL7349473 0.87 ALDH1A1 (0.50) ALDH1A1KDM4ELMNAHSD17B10PARP1
SCHEMBL7342194 0.83 ALDH1A1 (0.65) ALDH1A1KDM4ELMNAHSD17B10PARP1
SCHEMBL7345653 0.83 PARP1 (0.46) ALDH1A1KDM4ELMNAPARP1MAPT
SCHEMBL7338765 0.78 KDM4E (0.51) ALDH1A1KDM4ELMNAHSD17B10PARP1
SCHEMBL7341095 0.78 DAO (0.61) ALDH1A1KDM4ELMNAHSD17B10PARP1
SCHEMBL7339379 0.78 PARP1 (0.57) ALDH1A1KDM4ELMNAHSD17B10PARP1
SCHEMBL7349477 0.75 KDM4E (0.51) ALDH1A1KDM4ELMNAHSD17B10PARP1
SCHEMBL4459257 0.73 HSD17B10 (0.73) ALDH1A1KDM4ELMNAHSD17B10PARP1
SCHEMBL11095481 0.71 PARP1 (0.54) ALDH1A1KDM4ELMNAPARP1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4511569-A Tricyclic lactams and derivatives useful in increasing cardiac contractility SCHERING CORPORATION (US) 1985-04-16 US disclosed
EP-0102046-A1 Tricyclic lactams, method for making them, pharmaceutical compositions containing them SCHERING CORPORATION (US) 1984-03-07 EP disclosed