SCHEMBL11099683

SCHEMBL11099683

COc1cc(NC(C)=O)c(Cl)cc1NC(=O)C1CC2CCC(C1)N2Cc1cccs1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.45
CYP2C19 P33261 1/20 0.45
KMT2A Q03164 6/20 0.45
MEN1 O00255 5/20 0.45
TDP1 Q9NUW8 3/20 0.45
LMNA P02545 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
OPRM1 P35372 1/20 0.44
OPRK1 P41145 1/20 0.44
KCNH2 Q12809 1/20 0.44
TSHR P16473 1/20 0.42
APOBEC3A P31941 1/20 0.42
APOBEC3G Q9HC16 1/20 0.42
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
POLB P06746 1/20 0.41
MAPT P10636 1/20 0.41
THRB P10828 1/20 0.41
RECQL P46063 1/20 0.41
BLM P54132 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11100155 0.90 OPRM1 (0.45) CYP2D6CYP2C19KMT2AMEN1TDP1
SCHEMBL11097106 0.89 DRD2 (0.47) CYP2D6CYP2C19KMT2AMEN1TDP1
SCHEMBL11099128 0.86 MEN1 (0.52) CYP2D6CYP2C19KMT2AMEN1LMNA
SCHEMBL11092131 0.86 DRD4 (0.51) KMT2AMEN1TSHRDRD4DRD3
SCHEMBL11097236 0.86 MAPT (0.45) CYP2D6CYP2C19KMT2AMEN1TDP1
SCHEMBL11096164 0.84 CXCR6 (0.48) TSHRDRD4DRD3DRD2
SCHEMBL11092436 0.84 MEN1 (0.51) KMT2AMEN1OPRM1OPRK1KCNH2
SCHEMBL11270191 0.84 CXCR4 (0.47) CYP2D6CYP2C19KMT2AMEN1LMNA
SCHEMBL11098468 0.83 TSHR (0.44) TSHRDRD4DRD3DRD2
SCHEMBL11096744 0.80 UBE2M (0.45) KMT2AMEN1LMNAALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0031219-B1 ANILINE DERIVATIVES BEECHAM GROUP PLC (GB) 1984-03-07 EP disclosed
US-4350691-A ANTIEMETICS BEECHAM GROUP LIMITED (GB) 1982-09-21 US disclosed
EP-0031219-A1 Aniline derivatives BEECHAM GROUP PLC (GB) 1981-07-01 EP disclosed