SCHEMBL11270191

SCHEMBL11270191

COc1ccc(CN2C3CCC2CC(C(=O)Nc2cc(Cl)c(NC(C)=O)cc2OC)C3)cc1

nearest known ligand 0.51

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CXCR4 P61073 1/20 0.47
TSHR P16473 1/20 0.45
L3MBTL1 Q9Y468 2/20 0.44
LTA4H P09960 1/20 0.44
ALPL P05186 1/20 0.43
ALPI P09923 1/20 0.43
ALPG P10696 1/20 0.43
CCR1 P32246 1/20 0.43
DRD4 P21917 5/20 0.43
DRD3 P35462 3/20 0.43
DRD2 P14416 2/20 0.43
CYP2D6 P10635 1/20 0.42
CYP2C19 P33261 1/20 0.42
DRD5 P21918 1/20 0.42
MEN1 O00255 1/20 0.42
LMNA P02545 1/20 0.42
MAPT P10636 1/20 0.42
KMT2A Q03164 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11096164 0.93 CXCR6 (0.48) TSHRCCR1DRD4DRD3DRD2
SCHEMBL11092436 0.93 MEN1 (0.51) TSHRCCR1DRD4DRD3DRD2
SCHEMBL11098468 0.92 TSHR (0.44) TSHRCCR1DRD4DRD3DRD2
SCHEMBL11092131 0.91 DRD4 (0.51) TSHRDRD4DRD3DRD2DRD5
SCHEMBL11270864 0.89 CXCR4 (0.46) CXCR4TSHRL3MBTL1LTA4HALPL
SCHEMBL11097949 0.88 DRD2 (0.51) CXCR4TSHRL3MBTL1LTA4HALPL
SCHEMBL11089660 0.85 HCRTR1 (0.53) CXCR4TSHRMEN1MAPTKMT2A
SCHEMBL11097656 0.84 CXCR4 (0.45) CXCR4TSHRL3MBTL1LTA4HALPL
SCHEMBL11096744 0.84 UBE2M (0.45) DRD4DRD3DRD2DRD5MEN1
SCHEMBL11099683 0.84 CYP2D6 (0.45) TSHRL3MBTL1ALPLALPIALPG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0031219-A1 Aniline derivatives BEECHAM GROUP PLC (GB) 1981-07-01 EP claimed
US-4350691-A ANTIEMETICS BEECHAM GROUP LIMITED (GB) 1982-09-21 US disclosed
EP-0031219-A1 Aniline derivatives BEECHAM GROUP PLC (GB) 1981-07-01 EP disclosed