SCHEMBL11099776

SCHEMBL11099776

COc1ccc(C(C#N)(CCC(=O)O)CCC(=O)O)cc1Br

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 2/20 0.51
CASP1 P29466 1/20 0.51
ALDH1A1 P00352 3/20 0.42
CYP2C9 P11712 1/20 0.42
TSHR P16473 1/20 0.42
HIF1A Q16665 1/20 0.42
HPGD P15428 3/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C19 P33261 1/20 0.41
L3MBTL1 Q9Y468 2/20 0.40
HTT P42858 1/20 0.38
KLKB1 P03952 1/20 0.38
PPARA Q07869 3/20 0.37
PPARD Q03181 1/20 0.37
MEN1 O00255 1/20 0.36
LMNA P02545 1/20 0.36
KMT2A Q03164 1/20 0.36
KDM4E B2RXH2 1/20 0.36
TDP1 Q9NUW8 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7384417 0.88 HSD17B10 (0.66) HSD17B10CASP1ALDH1A1HPGDCYP1A2
SCHEMBL7421932 0.81 CASP1 (0.53) HSD17B10CASP1ALDH1A1CYP2C9L3MBTL1
SCHEMBL7424415 0.80 CASP1 (0.50) HSD17B10CASP1L3MBTL1
SCHEMBL11830247 0.79 CASP1 (0.54) HSD17B10CASP1ALDH1A1CYP2C9TSHR
SCHEMBL11091478 0.78 NPC1 (0.46) HSD17B10CASP1ALDH1A1HPGDCYP1A2
SCHEMBL5703639 0.78 PDE4B (0.50) HSD17B10CASP1
SCHEMBL11830796 0.78 MAPT (0.38) HSD17B10CASP1ALDH1A1CYP2C9TSHR
SCHEMBL11099780 0.78 HDAC1 (0.43) HSD17B10ALDH1A1TSHRHPGDCYP1A2
SCHEMBL7375552 0.76 HSD17B10 (0.64) HSD17B10CASP1ALDH1A1TSHRCYP1A2
SCHEMBL11074467 0.76 LMNA (0.46) HSD17B10CASP1ALDH1A1HPGDCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4460604-A ANALGESICS, NARCOTIC ANTAGONIST THE UPJOHN COMPANY (US) 1984-07-17 US disclosed
US-4180584-A ANALGESIC; NARCOTIC ANTAGONIST THE UPJOHN COMPANY (US) 1979-12-25 US disclosed
US-4065573-A ANALGESICS THE UPJOHN COMPANY (US) 1977-12-27 US disclosed