SCHEMBL11111875

SCHEMBL11111875

COc1ccc(Cl)cc1C1(C#N)CCN(S(=O)(=O)c2ccc(C)cc2)CC1

nearest known ligand 0.50

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.50
LMNA P02545 4/20 0.50
MEN1 O00255 4/20 0.50
KMT2A Q03164 4/20 0.50
MAPK1 P28482 2/20 0.50
HSD17B10 Q99714 2/20 0.50
SMN1; SMN2 Q16637 2/20 0.48
TSHR P16473 2/20 0.48
GAA P10253 1/20 0.48
KDM4E B2RXH2 3/20 0.47
MAPT P10636 1/20 0.45
POLB P06746 2/20 0.45
HPGD P15428 1/20 0.45
RAB9A P51151 1/20 0.45
HTT P42858 2/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
STAT3 P40763 1/20 0.44
KCNT1 Q5JUK3 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11117214 0.86 HTT (0.51) ALDH1A1LMNAMEN1KMT2ASMN1; SMN2
SCHEMBL11118953 0.85 ADRA1D (0.53) ALDH1A1LMNAMEN1KMT2ATSHR
SCHEMBL11121167 0.81 CYP2C19 (0.57) ALDH1A1LMNAMEN1KMT2AMAPK1
SCHEMBL11114004 0.81 ALDH1A1 (0.52) ALDH1A1LMNAMEN1KMT2AMAPK1
SCHEMBL11602090 0.80 OPRM1 (0.56) ALDH1A1LMNAMEN1KMT2AHSD17B10
SCHEMBL11124896 0.79 OXTR (0.55) ALDH1A1LMNAMEN1KMT2ASMN1; SMN2
SCHEMBL11113941 0.78 SMN1; SMN2 (0.52) ALDH1A1LMNAMEN1KMT2AMAPK1
SCHEMBL11178032 0.77 OXTR (0.50) ALDH1A1LMNAMEN1KMT2ASMN1; SMN2
SCHEMBL5470612 0.74 KMT2A (0.62) LMNAMEN1KMT2AMAPTPOLB
SCHEMBL11115677 0.74 OXTR (0.55) ALDH1A1LMNAMEN1KMT2ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0034415-B1 1-(CYCLOHEXYL OR CYCLOHEXENYL)-4-ARYL-4-PIPERIDINECARBOXYLIC ACID DERIVATIVES JANSSEN PHARMACEUTICA N.V. (BE) 1984-05-30 EP disclosed
US-4369184-A ANTIHISTAMINES; HETEROCYCLIC NITRILES JANSSEN PHARMACEUTICA N.V. (BE) 1983-01-18 US disclosed
EP-0034415-A1 1-(Cyclohexyl or cyclohexenyl)-4-aryl-4-piperidinecarboxylic acid derivatives JANSSEN PHARMACEUTICA N.V. (BE) 1981-08-26 EP disclosed