SCHEMBL11113464

SCHEMBL11113464

COc1ccc(C(=O)N(C)CCN(C)CCC(c2ccccc2)c2ccccc2)cc1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 1/20 0.63
PTGDR2 Q9Y5Y4 1/20 0.50
SLC6A9 P48067 1/20 0.49
TDP1 Q9NUW8 1/20 0.49
ALDH1A1 P00352 3/20 0.48
MAPT P10636 3/20 0.48
HPGD P15428 3/20 0.47
KDM4E B2RXH2 1/20 0.47
LMNA P02545 2/20 0.47
POLB P06746 1/20 0.47
GAA P10253 1/20 0.47
PKM P14618 1/20 0.47
RECQL P46063 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
CNR1 P21554 1/20 0.46
CNR2 P34972 1/20 0.46
ACHE P22303 1/20 0.46
MEN1 O00255 4/20 0.46
KMT2A Q03164 4/20 0.46
NPC1 O15118 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11111247 0.85 CDK4 (0.46) DRD2SLC6A9LMNACNR1NPSR1
SCHEMBL11116808 0.83 DRD2 (0.45) DRD2SLC6A9ALDH1A1MAPTKDM4E
SCHEMBL9117039 0.81 MEN1 (0.59) PTGDR2TDP1ALDH1A1MAPTHPGD
SCHEMBL19479112 0.80 DRD2 (0.74) DRD2ALDH1A1MAPTHPGDKDM4E
SCHEMBL11130111 0.78 TSHR (0.57) SLC6A9TDP1ALDH1A1MAPTHPGD
SCHEMBL19479124 0.78 DRD2 (1.00) DRD2MAPTACHEMEN1KMT2A
SCHEMBL11110461 0.76 TSHR (0.59) TDP1ALDH1A1MAPTHPGDLMNA
SCHEMBL13181408 0.76 MLYCD (0.64) DRD2MAPTHPGDKDM4EACHE
SCHEMBL16941089 0.76 DRD2 (0.59) DRD2ALDH1A1MAPTHPGDKDM4E
SCHEMBL11115848 0.74 SIGMAR1 (0.55) SLC6A9ALDH1A1MAPTHPGDLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0041757-B1 ETHYLENDIAMINE DERIVATIVES, PREPARATION THEREOF, PHARMACEUTICAL COMPOSITIONS CONTAINING SAME AND INTERMEDIATES FOR THEIR PREPARATION Simes S.p.A. (IT) 1984-11-07 EP disclosed
EP-0041757-A1 Ethylendiamine derivatives, preparation thereof, pharmaceutical compositions containing same and intermediates for their preparation Simes S.p.A. (IT) 1981-12-16 EP disclosed