SCHEMBL11110461

SCHEMBL11110461

COc1ccc(C(CCN(C)CCN(C)Cc2ccccc2)c2ccccc2)cc1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.59
TDP1 Q9NUW8 1/20 0.50
ACHE P22303 1/20 0.50
ALDH1A1 P00352 3/20 0.49
MAPT P10636 3/20 0.49
MEN1 O00255 4/20 0.49
KMT2A Q03164 4/20 0.49
SIGMAR1 Q99720 2/20 0.48
LMNA P02545 2/20 0.47
HPGD P15428 2/20 0.47
POLB P06746 1/20 0.47
GAA P10253 1/20 0.47
PKM P14618 1/20 0.47
RECQL P46063 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
NPC1 O15118 1/20 0.47
TP53 P04637 1/20 0.47
HTT P42858 1/20 0.47
RAB9A P51151 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11130111 0.96 TSHR (0.57) TSHRTDP1ACHEALDH1A1MAPT
SCHEMBL9750655 0.88 HTR2A (0.58) TSHRALDH1A1SIGMAR1LMNASMN1; SMN2
SCHEMBL8297797 0.85 HTR2A (0.62) TSHRALDH1A1SIGMAR1LMNASMN1; SMN2
SCHEMBL11115848 0.81 SIGMAR1 (0.55) ALDH1A1MAPTMEN1KMT2ASIGMAR1
SCHEMBL9750783 0.78 ALDH1A1 (0.51) ALDH1A1MAPTMEN1KMT2ASIGMAR1
SCHEMBL11115510 0.78 ALDH1A1 (0.58) ACHEALDH1A1MAPTMEN1KMT2A
SCHEMBL11114924 0.78 SIGMAR1 (0.51) TSHRSIGMAR1L3MBTL1HTR2AHRH1
SCHEMBL11115618 0.78 HRH1 (0.50) TSHRMAPTMEN1KMT2ASIGMAR1
SCHEMBL16039094 0.77 ACHE (0.76) TSHRACHEMAPTMEN1KMT2A
SCHEMBL11113464 0.76 DRD2 (0.63) TDP1ACHEALDH1A1MAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0041757-B1 ETHYLENDIAMINE DERIVATIVES, PREPARATION THEREOF, PHARMACEUTICAL COMPOSITIONS CONTAINING SAME AND INTERMEDIATES FOR THEIR PREPARATION Simes S.p.A. (IT) 1984-11-07 EP disclosed
EP-0041757-A1 Ethylendiamine derivatives, preparation thereof, pharmaceutical compositions containing same and intermediates for their preparation Simes S.p.A. (IT) 1981-12-16 EP disclosed