SCHEMBL11114414

SCHEMBL11114414

COc1ccccc1C1(C(=O)O)CCN(S(=O)(=O)c2ccc(C)cc2)CC1

nearest known ligand 0.69

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 2/20 0.69
KMT2A Q03164 3/20 0.58
GAA P10253 4/20 0.56
MEN1 O00255 2/20 0.56
OXTR P30559 1/20 0.55
CYP2D6 P10635 2/20 0.52
PKM P14618 1/20 0.52
ALDH1A1 P00352 2/20 0.50
LMNA P02545 1/20 0.50
HTT P42858 1/20 0.50
GFER P55789 1/20 0.50
TSHR P16473 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
USP2 O75604 1/20 0.50
CYP3A4 P08684 1/20 0.50
CYP2C9 P11712 1/20 0.50
KDM4E B2RXH2 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11120207 0.90 CYP2C19 (0.58) CYP2C19KMT2AGAAMEN1OXTR
SCHEMBL11118092 0.87 CYP2C19 (0.55) CYP2C19KMT2AGAAMEN1OXTR
SCHEMBL11121167 0.85 CYP2C19 (0.57) CYP2C19KMT2AGAAMEN1ALDH1A1
SCHEMBL11117181 0.81 CYP2C19 (0.67) CYP2C19KMT2AGAAMEN1OXTR
SCHEMBL11118953 0.80 ADRA1D (0.53) CYP2C19KMT2AGAAMEN1OXTR
SCHEMBL11128806 0.77 CYP2C19 (0.62) CYP2C19KMT2AGAAMEN1OXTR
SCHEMBL11127656 0.77 CYP2C19 (0.62) CYP2C19KMT2AGAAMEN1OXTR
SCHEMBL2699791 0.76 KMT2A (0.76) CYP2C19KMT2AMEN1CYP2D6PKM
SCHEMBL11114004 0.76 ALDH1A1 (0.52) CYP2C19KMT2AGAAMEN1ALDH1A1
SCHEMBL3443849 0.76 L3MBTL1 (0.51) KMT2AMEN1ALDH1A1LMNAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0034415-B1 1-(CYCLOHEXYL OR CYCLOHEXENYL)-4-ARYL-4-PIPERIDINECARBOXYLIC ACID DERIVATIVES JANSSEN PHARMACEUTICA N.V. (BE) 1984-05-30 EP disclosed
US-4369184-A ANTIHISTAMINES; HETEROCYCLIC NITRILES JANSSEN PHARMACEUTICA N.V. (BE) 1983-01-18 US disclosed