SCHEMBL11119745

SCHEMBL11119745

CCN(CC)CCCNC1c2ccccc2COc2ccc(F)cc21

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.39
ALOX15 P16050 1/20 0.39
TBXAS1 P24557 1/20 0.37
MAPK14 Q16539 1/20 0.36
BCHE P06276 1/20 0.36
ACHE P22303 1/20 0.36
SLC6A2 P23975 3/20 0.35
SLC6A4 P31645 3/20 0.35
HTR2C P28335 3/20 0.35
SLC6A3 Q01959 2/20 0.35
HTR2B P41595 1/20 0.35
DRD2 P14416 2/20 0.34
DRD3 P35462 2/20 0.34
CHRM1 P11229 1/20 0.34
ADRA2C P18825 1/20 0.34
HTR2A P28223 1/20 0.34
ADRA1A P35348 1/20 0.34
HRH1 P35367 1/20 0.34
OPRM1 P35372 1/20 0.34
OPRK1 P41145 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11129673 0.93 TBXAS1 (0.38) ALDH1A1ALOX15TBXAS1MAPK14SLC6A2
SCHEMBL11115157 0.89 HTR2B (0.43) TBXAS1SLC6A2SLC6A4HTR2CSLC6A3
SCHEMBL11111420 0.88 ALOX15 (0.40) ALDH1A1ALOX15TBXAS1BCHEACHE
SCHEMBL11113367 0.87 ALDH1A1 (0.39) ALDH1A1ALOX15TBXAS1BCHEACHE
SCHEMBL11114001 0.87 MEN1 (0.40) ALDH1A1ALOX15TBXAS1BCHEACHE
SCHEMBL11112434 0.85 SMPD1 (0.45) ALDH1A1ALOX15TBXAS1HTR2BDRD2
SCHEMBL11117688 0.84 HTR2B (0.44) ALDH1A1TBXAS1MAPK14SLC6A2SLC6A4
SCHEMBL10999576 0.83 TBXAS1 (0.46) ALDH1A1ALOX15TBXAS1HTR2CSLC6A3
SCHEMBL11114115 0.81 TBXAS1 (0.39) ALDH1A1ALOX15TBXAS1SLC6A2HTR2C
SCHEMBL11112746 0.80 TBXAS1 (0.43) TBXAS1SLC6A2SLC6A4HTR2CHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0038564-B1 DIBENZ (B,E) OXEPIN DERIVATIVES AND PHARMACEUTICAL COMPOSITIONS COMPRISING THEM KYOWA HAKKO KOGYO CO., LTD (JP) 1984-09-12 EP disclosed
US-4396550-A ANTICHOLINERGIC, ANTIHISTIMINIC AGENTS KYOWA HAKKO KOGYO CO., LTD. (JP) 1983-08-02 US disclosed
EP-0038564-A1 Dibenz (b,e) oxepin derivatives and pharmaceutical compositions comprising them KYOWA HAKKO KOGYO CO., LTD (JP) 1981-10-28 EP disclosed