SCHEMBL1114522

SCHEMBL1114522

Oc1c(Cl)cc(C2=NCON2Cc2cccc(C(F)(F)F)c2)cc1Cl

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.41
KDM4E B2RXH2 1/20 0.41
GAA P10253 1/20 0.41
HTT P42858 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
P2RX7 Q99572 1/20 0.39
S1PR1 P21453 1/20 0.39
S1PR5 Q9H228 1/20 0.39
POLB P06746 1/20 0.38
LMNA P02545 2/20 0.38
HSD17B13 Q7Z5P4 1/20 0.37
MEN1 O00255 1/20 0.37
PLA2G1B P04054 1/20 0.37
HPGD P15428 1/20 0.37
KMT2A Q03164 1/20 0.37
GFER P55789 1/20 0.37
FAAH O00519 1/20 0.37
AKR1C3 P42330 1/20 0.37
AKR1C2 P52895 1/20 0.37
ICMT O60725 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1114402 0.87 ALDH1A1 (0.41) ALDH1A1KDM4EGAAHTTL3MBTL1
SCHEMBL1114336 0.79 KDM4E (0.39) ALDH1A1KDM4EGAAHTTP2RX7
SCHEMBL1114224 0.76 KDM4E (0.41) ALDH1A1KDM4EGAAHTTL3MBTL1
SCHEMBL1114553 0.74 MGLL (0.39) ALDH1A1LMNAFAAHAKR1C3
SCHEMBL1114223 0.70 P2RX7 (0.39) ALDH1A1KDM4EGAAHTTL3MBTL1
SCHEMBL1114525 0.67 P2RX7 (0.39) ALDH1A1KDM4EGAAHTTL3MBTL1
SCHEMBL4351774 0.65 FFAR1 (0.54) ALDH1A1GAAL3MBTL1P2RX7LMNA
SCHEMBL1114208 0.64 KDM4E (0.36) ALDH1A1KDM4E
SCHEMBL28160828 0.61 POLB (0.54) ALDH1A1KDM4EGAAHTTL3MBTL1
SCHEMBL17159726 0.61 POLB (0.54) ALDH1A1KDM4EGAAHTTL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2278879-A2 COMPOUNDS, COMPOSITIONS AND METHODS COMPRISING OXADIAZOLE DERIVATIVES Institute for OneWorld Health (US) 2011-02-02 EP claimed
WO-2009131957-A2 COMPOUNDS, COMPOSITIONS AND METHODS COMPRISING OXADIAZOLE DERIVATIVES INSTITUTE FOR ONEWORLD HEALTH (US) 2009-10-29 WO claimed
EP-2278879-A2 COMPOUNDS, COMPOSITIONS AND METHODS COMPRISING OXADIAZOLE DERIVATIVES Institute for OneWorld Health (US) 2011-02-02 EP disclosed
WO-2009131957-A2 COMPOUNDS, COMPOSITIONS AND METHODS COMPRISING OXADIAZOLE DERIVATIVES INSTITUTE FOR ONEWORLD HEALTH (US) 2009-10-29 WO disclosed