SCHEMBL1114749

SCHEMBL1114749

Oc1c(Cl)cc(C2=NCN(Cc3cccc(OC(F)(F)F)c3)O2)cc1Cl

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HSD17B13 Q7Z5P4 2/20 0.40
KCNN3 Q9UGI6 1/20 0.38
ACLY P53396 1/20 0.37
CETP P11597 2/20 0.37
DRD4 P21917 1/20 0.37
FEN1 P39748 1/20 0.37
ROCK2 O75116 1/20 0.37
ROCK1 Q13464 1/20 0.37
KCNN4 O15554 4/20 0.37
GRIN2B Q13224 1/20 0.36
P2RX7 Q99572 1/20 0.36
AMPD2 Q01433 1/20 0.36
ATM Q13315 1/20 0.36
DRD2 P14416 1/20 0.36
DRD1 P21728 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1114292 0.88 MEP1B (0.36) CETPROCK2P2RX7
SCHEMBL1114224 0.84 KDM4E (0.41) HSD17B13P2RX7
SCHEMBL1114208 0.79 KDM4E (0.36)
SCHEMBL4516945 0.73 HSD17B13 (0.42) HSD17B13KCNN3FEN1KCNN4P2RX7
SCHEMBL1114748 0.69 HSD17B13 (0.40) HSD17B13KCNN3CETPDRD4FEN1
SCHEMBL3240176 0.67 RXRA (0.43) FEN1ROCK2ROCK1GRIN2BP2RX7
SCHEMBL4504413 0.66 FEN1 (0.39) HSD17B13CETPDRD4FEN1KCNN4
SCHEMBL1114303 0.65 MEP1B (0.36) CETPROCK2P2RX7
SCHEMBL690748 0.65 ROCK2 (0.52) ROCK2ROCK1
SCHEMBL28160866 0.63 KCNN3 (0.46) KCNN3DRD4ROCK2ROCK1KCNN4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2278879-A2 COMPOUNDS, COMPOSITIONS AND METHODS COMPRISING OXADIAZOLE DERIVATIVES Institute for OneWorld Health (US) 2011-02-02 EP claimed
WO-2009131957-A2 COMPOUNDS, COMPOSITIONS AND METHODS COMPRISING OXADIAZOLE DERIVATIVES INSTITUTE FOR ONEWORLD HEALTH (US) 2009-10-29 WO claimed