SCHEMBL11180

SCHEMBL11180

CCOC(=O)C1(c2ccc(-c3ccccc3)c(-c3onc(C)c3CN3CCCC(c4ccccc4)C3)c2)CC1

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 4/20 0.38
OPRD1 P41143 3/20 0.38
OPRK1 P41145 3/20 0.38
DGAT2 Q96PD7 1/20 0.38
ATM Q13315 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
SIGMAR1 Q99720 5/20 0.37
HSD11B1 P28845 1/20 0.37
LMNA P02545 1/20 0.37
TSHR P16473 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
SLC22A1 O15245 1/20 0.36
SLC6A4 P31645 1/20 0.36
ADRA1A P35348 1/20 0.36
KCNH2 Q12809 1/20 0.36
KCNA3 P22001 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11688 0.95 SIGMAR1 (0.40) OPRM1OPRD1OPRK1SIGMAR1SLC22A1
SCHEMBL11181 0.93 OPRM1 (0.42) OPRM1OPRD1OPRK1ATML3MBTL1
SCHEMBL11879 0.92 SIGMAR1 (0.42) OPRM1OPRD1OPRK1SIGMAR1NPSR1
SCHEMBL11689 0.88 OPRM1 (0.43) OPRM1OPRD1OPRK1SIGMAR1SLC22A1
SCHEMBL5236 0.88 OPRM1 (0.43) OPRM1OPRD1OPRK1ATML3MBTL1
SCHEMBL11880 0.84 SIGMAR1 (0.46) OPRM1OPRD1OPRK1SIGMAR1SLC22A1
SCHEMBL4483 0.84 OPRM1 (0.45) OPRM1OPRD1OPRK1SIGMAR1SLC22A1
SCHEMBL10120 0.81 OPRM1 (0.43) OPRM1OPRD1OPRK1LMNATSHR
SCHEMBL4330 0.80 SIGMAR1 (0.47) OPRM1OPRD1OPRK1SIGMAR1SLC22A1
SCHEMBL4729 0.79 HSD11B1 (0.45) ATML3MBTL1HSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2483251-A2 POLYCYCLIC COMPOUNDS AS LYSOPHOSPHATIDIC ACID RECEPTOR ANTAGONISTS Amira Pharmaceuticals, Inc. (US) 2012-08-08 EP disclosed
WO-2011041462-A2 POLYCYCLIC COMPOUNDS AS LYSOPHOSPHATIDIC ACID RECEPTOR ANTAGONISTS AMIRA PHARMACEUTICALS, INC. (US) 2011-04-07 WO disclosed