SCHEMBL11201464

SCHEMBL11201464

COc1ccc(C(O)c2cccc(C(F)(F)F)c2)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.54
MEN1 O00255 2/20 0.54
PNMT P11086 1/20 0.49
MAPT P10636 2/20 0.48
ALDH1A1 P00352 1/20 0.48
GAA P10253 1/20 0.48
TDP1 Q9NUW8 1/20 0.48
MAOB P27338 1/20 0.47
CES2 O00748 1/20 0.46
ACP3 P15309 1/20 0.46
POLB P06746 2/20 0.45
LMNA P02545 1/20 0.45
HTT P42858 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
NR1H4 Q96RI1 1/20 0.44
KDM4E B2RXH2 1/20 0.43
BACE1 P56817 1/20 0.43
GRIN2B Q13224 1/20 0.43
IDO1 P14902 1/20 0.43
TDO2 P48775 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6473252 0.85 CASR (0.50) KMT2AMEN1MAPTTDP1ACP3
SCHEMBL10552240 0.85 CASR (0.51) KMT2AMEN1ALDH1A1TDP1SMN1; SMN2
SCHEMBL5782693 0.84 MEN1 (0.58) KMT2AMEN1ALDH1A1TDP1MAOB
SCHEMBL4135956 0.83 PNMT (0.65) PNMTMAPTALDH1A1CES2ACP3
SCHEMBL4135655 0.82 PNMT (0.59) KMT2AMEN1PNMTMAPTALDH1A1
SCHEMBL11193839 0.82 ALDH1A1 (0.48) KMT2AMEN1PNMTMAPTALDH1A1
SCHEMBL2010410 0.82 IDO1 (0.47) KMT2AMEN1PNMTMAPTALDH1A1
SCHEMBL10889071 0.81 PNMT (0.54) KMT2AMEN1PNMTMAPTALDH1A1
Hydrochloric Acid SCHEMBL2013413 0.81 IDO1 (0.49) KMT2AMEN1PNMTMAPTALDH1A1
SCHEMBL28519052 0.79 MEN1 (0.51) KMT2AMEN1MAPTTDP1MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4377578-A ANTIANAPHYLACTIC AGENTS, ANTIHISTAMINES JANSSEN PHARMACEUTICA, N.V. (BE) 1983-03-22 US disclosed
US-4250176-A BENZIMIDAZOLE-2-ONE, BENZOTHIAZOL-2-ONE, OR BENZOXAZOL-2-ONE SUBSTITUTIONS, ANTIANAPHALACTIC AGENTS, ANTIHISTAMINES JANSSEN PHARMACEUTICA N.V. (BE) 1981-02-10 US disclosed
US-4200641-A ANTIANAPHYLACTIC AGENTS, ANTIHISTAMINES JANSSEN PHARMACEUTICA, N.V. (BE) 1980-04-29 US disclosed