SCHEMBL11201872

SCHEMBL11201872

Nc1nc(N2CCN(Cc3ccccc3)CC2)nc2sccc12

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.53
HTR2C P28335 4/20 0.50
HTR3A P46098 3/20 0.50
HTR3E A5X5Y0 2/20 0.50
HTR3B O95264 2/20 0.50
HTR1A P08908 2/20 0.50
HTR3D Q70Z44 2/20 0.50
HTR3C Q8WXA8 2/20 0.50
CASP1 P29466 1/20 0.50
CASP5 P51878 1/20 0.50
HRH4 Q9H3N8 1/20 0.47
HTT P42858 2/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
KDM4E B2RXH2 3/20 0.46
MAPT P10636 3/20 0.46
NPSR1 Q6W5P4 2/20 0.46
MAPK1 P28482 1/20 0.46
ADORA2A P29274 1/20 0.46
MC4R P32245 1/20 0.46
LMNA P02545 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1083795 0.81 HTR3A (0.68) GAAHTR3ACASP1CASP5HRH4
SCHEMBL17377841 0.81 HTR3E (0.56) GAAHTR2CHTR3AHTR3EHTR3B
SCHEMBL11201044 0.75 HTR2C (0.70) HTR2CHTR3ACASP1CASP5HRH4
SCHEMBL16164244 0.72 HTT (0.68) GAAHTR2CHTR3AHTR3EHTR3B
SCHEMBL11384876 0.72 CASP1 (0.66) GAACASP1CASP5HTTSMN1; SMN2
SCHEMBL11282875 0.72 LMNA (0.58) GAACASP1CASP5HTTSMN1; SMN2
SCHEMBL11278102 0.72 LMNA (0.56) GAACASP1CASP5HTTSMN1; SMN2
SCHEMBL11201579 0.71 MEN1 (0.50) GAAHTR1AHTTSMN1; SMN2KDM4E
Hydrochloric Acid SCHEMBL7834533 0.71 NSD2 (0.65) GAAKDM4E
Hydrochloric Acid SCHEMBL7834531 0.71 NSD2 (0.65) GAAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0082023-A2 Thienopyrimidine derivatives, their preparation and their medical use SANKYO COMPANY LIMITED (JP) 1983-06-22 EP disclosed