SCHEMBL1120580

SCHEMBL1120580

CCOC(=O)CNNc1cccnc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.48
MAPT P10636 2/20 0.48
NPC1 O15118 2/20 0.48
RAB9A P51151 2/20 0.48
PKM P14618 1/20 0.48
TSHR P16473 1/20 0.46
KDM4E B2RXH2 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
RXFP1 Q9HBX9 1/20 0.45
NCOA1 Q15788 1/20 0.45
NCOA3 Q9Y6Q9 1/20 0.45
LMNA P02545 2/20 0.44
POLB P06746 2/20 0.44
TBXAS1 P24557 1/20 0.44
NAMPT P43490 2/20 0.44
NOTUM Q6P988 2/20 0.44
TRPV1 Q8NER1 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2C19 P33261 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7362493 0.85 RAB9A (0.50) ALDH1A1MAPTNPC1RAB9APKM
SCHEMBL9641365 0.80 ALDH1A1 (0.51) ALDH1A1MAPTNPC1RAB9APKM
SCHEMBL25528963 0.78 LMNA (0.58) ALDH1A1MAPTNPC1RAB9APKM
SCHEMBL7364359 0.77 TOP2A (0.51) ALDH1A1MAPTNPC1RAB9APKM
SCHEMBL1120518 0.77 GAA (0.53) ALDH1A1MAPTNPC1RAB9ATSHR
SCHEMBL966665 0.76 NPC1 (0.59) ALDH1A1MAPTNPC1RAB9APKM
SCHEMBL30058651 0.76 NPC1 (0.59) ALDH1A1MAPTNPC1RAB9APKM
SCHEMBL1120545 0.75 GAA (0.57) ALDH1A1MAPTNPC1RAB9ATSHR
SCHEMBL714353 0.74 THRB (0.63) ALDH1A1MAPTNPC1RAB9AKDM4E
SCHEMBL1120688 0.74 MAPT (0.59) ALDH1A1MAPTNPC1RAB9ATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2280968-A2 PYRIDO [3, 4-B]INDOLES AND METHODS OF USE Medivation Technologies, Inc. (US) 2011-02-09 EP disclosed
WO-2009120717-A2 PYRIDO [3, 4-B] INDOLES AND METHODS OF USE MEDIVATION TECHNOLOGIES, INC. (US) 2009-10-01 WO disclosed