SCHEMBL11208244

SCHEMBL11208244

COc1ccc([C@H](O)C(=O)OC(=O)[C@@H](C)N)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM8 O00222 1/20 0.44
GRM6 O15303 1/20 0.44
GRM4 Q14833 1/20 0.44
ALOX5 P09917 1/20 0.43
MEN1 O00255 1/20 0.43
RAB9A P51151 1/20 0.43
KMT2A Q03164 1/20 0.43
AOC3 Q16853 2/20 0.41
CA1 P00915 3/20 0.41
CA2 P00918 3/20 0.41
PARP1 P09874 1/20 0.41
PARP10 Q53GL7 1/20 0.41
PARP2 Q9UGN5 1/20 0.41
PARP4 Q9UKK3 1/20 0.41
ACHE P22303 1/20 0.41
CYP1A2 P05177 2/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C19 P33261 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11208763 1.00 GRM8 (0.44) GRM8GRM6GRM4ALOX5MEN1
SCHEMBL8475304 0.90 CES2 (0.47) GRM8GRM6GRM4MEN1RAB9A
SCHEMBL11208359 0.83 ALOX5 (0.41) ALOX5KMT2AACHETDP1L3MBTL1
SCHEMBL11204316 0.83 ALOX5 (0.41) ALOX5KMT2AACHETDP1L3MBTL1
SCHEMBL11206228 0.82 GRIN2D (0.48) MEN1KMT2AAOC3CYP1A2CYP2D6
SCHEMBL11211253 0.82 GRIN2D (0.48) MEN1KMT2AAOC3CYP1A2CYP2D6
SCHEMBL9662942 0.81 NPSR1 (0.42) GRM8GRM6GRM4MEN1RAB9A
D-Alanine SCHEMBL11208761 0.80 GRM8 (0.49) GRM8GRM6GRM4ALOX5MEN1
Alanine SCHEMBL11205694 0.80 GRM8 (0.49) GRM8GRM6GRM4ALOX5MEN1
SCHEMBL14621033 0.80 AOC3 (0.46) GRM8GRM6GRM4ALOX5MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0009722-B1 OPTICALLY ACTIVE COMPLEX, ALANINE.RING-SUBSTITUTED MANDELIC ACID, AND THE METHOD FOR PRODUCING THE SAME NIPPON KAYAKU KABUSHIKI KAISHA (JP) 1983-03-02 EP claimed
EP-0009722-A1 Optically active complex, alanine.Ring-substituted mandelic acid, and the method for producing the same NIPPON KAYAKU KABUSHIKI KAISHA (JP) 1980-04-16 EP claimed