Fumaric Acid

Fumaric Acid

SCHEMBL11210787

CC(C)(CO)COC(=O)C(C)(C)CO.O=C(O)C=CC(=O)O

nearest known ligand 0.37

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Known targets — ChEMBL curated mechanism

ACEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ATP4AATP4BAXLBTKCACNA1CCACNA1DCACNA1FCACNA1SCCR5CHRM2CHRM3CPT1BCPT2DPP4DRD1DRD2EGFRERBB2ERBB4FLT3HRH1HRH3HTR1AHTR2AHTR2BHTR2CHTR4JAK1JAK2JAK3KCNH2KMT2AMAP2K1MAP2K2MEN1MLNRMPLMTORPPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PLK4PPARGRENS1PR1SLC6A2SLC6A3SLC6A4SMOTYK2atpAatpBatpCatpDatpEatpFatpFHatpGpol

The experimentally established mechanism targets of Fumaric Acid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 6/20 0.37
TSHR P16473 2/20 0.32
TP53 P04637 1/20 0.32
EGLN1 Q9GZT9 1/20 0.32
EGLN3 Q9H6Z9 1/20 0.32
CYP4F2 P78329 1/20 0.32
CYP4A11 Q02928 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26021 0.89 CYP4F2 (0.37) CYP4F2CYP4A11
Acrylic Acid SCHEMBL4622901 0.88 ALDH1A1 (0.38) TP53CYP4F2CYP4A11
SCHEMBL11210783 0.87 HCAR2 (0.44) HCAR2TP53
SCHEMBL12403725 0.85 CYP4F2 (0.35) CYP4F2CYP4A11
SCHEMBL27696058 0.83 ALDH1A1 (0.34) TP53CYP4F2CYP4A11
SCHEMBL12403723 0.82 CYP4F2 (0.38) TP53CYP4F2CYP4A11
SCHEMBL11805690 0.81 HCAR2 (0.53) HCAR2TSHRTP53EGLN1EGLN3
SCHEMBL3627793 0.81 HCAR2 (0.53) HCAR2TSHRTP53EGLN1EGLN3
Methacrylic Acid SCHEMBL6737902 0.81 CYP4F2 (0.31) CYP4F2CYP4A11
Acetoacetic Acid SCHEMBL9574542 0.79 KDM4E (0.31) CYP4F2CYP4A11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0020945-B1 COMPOSITIONS CONTAINING HALF ESTERS OF ORGANIC POLYOLS, A PROCESS FOR THEIR PRODUCTION AND USE OF THE COMPOSITIONS IN THE PRODUCTION OF MOULDED ARTICLES UNION CARBIDE CORPORATION (US) 1983-05-25 EP disclosed
US-4263413-A CURING ACRYLIC COPOLYMERS UNION CARBIDE CORPORATION (US) 1981-04-21 US disclosed