SCHEMBL11211367

SCHEMBL11211367

Cc1c(O)ccc(C(=O)c2ccc(O)cc2)c1O

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 5/20 0.56
HPGD P15428 4/20 0.56
ALDH1A1 P00352 4/20 0.56
HSD17B10 Q99714 3/20 0.56
LMNA P02545 2/20 0.56
KDM4E B2RXH2 2/20 0.56
RECQL P46063 2/20 0.56
TDP1 Q9NUW8 2/20 0.56
MAPK1 P28482 2/20 0.56
CYP3A4 P08684 1/20 0.56
LIG1 P18858 1/20 0.52
HTT P42858 3/20 0.50
ESR1 P03372 1/20 0.50
ESR2 Q92731 1/20 0.50
PKM P14618 1/20 0.50
ALOX15 P16050 2/20 0.47
MEN1 O00255 5/20 0.46
KMT2A Q03164 5/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
NPC1 O15118 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29215682 0.89 ALDH1A1 (0.54) MAPTHPGDALDH1A1HSD17B10LMNA
SCHEMBL11015751 0.87 LIG1 (0.53) MAPTHPGDALDH1A1HSD17B10LMNA
SCHEMBL25242597 0.86 KMT2A (0.56) MAPTHPGDALDH1A1HSD17B10LMNA
SCHEMBL30331291 0.85 MAPT (0.56) MAPTHPGDALDH1A1HSD17B10LMNA
SCHEMBL2859239 0.85 MAPT (0.56) MAPTHPGDALDH1A1HSD17B10LMNA
SCHEMBL1758260 0.84 KMT2A (0.51) MAPTHPGDALDH1A1HSD17B10KDM4E
SCHEMBL11218165 0.83 NPC1 (0.55) MAPTHPGDALDH1A1HSD17B10LMNA
SCHEMBL30506538 0.83 NPC1 (0.55) MAPTHPGDALDH1A1HSD17B10LMNA
SCHEMBL25251755 0.83 SIRT1 (0.57) MAPTHPGDALDH1A1HSD17B10LMNA
SCHEMBL29366288 0.82 HDAC1 (0.66) MAPTHPGDALDH1A1HSD17B10LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4349607-A UV Stabilizers, coating compositions and composite structures obtained therefrom GENERAL ELECTRIC COMPANY (US) 1982-09-14 US claimed
US-4288631-A 3-ALKYLHYDROXYBENZOPHENONES GENERAL ELECTRIC COMPANY (US) 1981-09-08 US claimed
US-10370349-B2 Functionalised benzopyran compounds and use thereof Kazia Therapeutics Limited (AU) 2019-08-06 US disclosed
US-20180141925-A1 FUNCTIONALISED BENZOPYRAN COMPOUNDS AND USE THEREOF Kazia Therapeutics Limited (AU) 2018-05-24 US disclosed
EP-2953938-B1 FUNCTIONALISED BENZOPYRAN COMPOUNDS AND USE THEREOF Novogen ltd (AU) 2017-08-02 EP disclosed
US-9701655-B2 Functionalised benzopyran compounds and use thereof NOVOGEN LIMITED (AU) 2017-07-11 US disclosed
US-20160340329-A1 FUNCTIONALISED BENZOPYRAN COMPOUNDS AND USE THEREOF VIVESTO AB (SE) 2016-11-24 US disclosed
EP-2953938-A1 FUNCTIONALISED BENZOPYRAN COMPOUNDS AND USE THEREOF Novogen Ltd. (AU) 2015-12-16 EP disclosed
WO-2015117202-A1 FUNCTIONALISED BENZOPYRAN COMPOUNDS AND USE THEREOF NOVOGEN LIMITED (AU) 2015-08-13 WO disclosed
US-4349607-A UV Stabilizers, coating compositions and composite structures obtained therefrom GENERAL ELECTRIC COMPANY (US) 1982-09-14 US disclosed
US-4288631-A 3-ALKYLHYDROXYBENZOPHENONES GENERAL ELECTRIC COMPANY (US) 1981-09-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20180141925-A1 FUNCTIONALISED BENZOPYRAN COMPOUNDS AND USE THEREOF BRCA1, BRAP, EP300 MAPT 704/4885HPGD 1157/4885ALDH1A1 298/4885
US-20160340329-A1 FUNCTIONALISED BENZOPYRAN COMPOUNDS AND USE THEREOF BRCA1, VHL, NQO1 MAPT 4629/4885HPGD 56/4885ALDH1A1 189/4885
US-10370349-B2 Functionalised benzopyran compounds and use thereof BRCA1, BRAP, EP300 MAPT 704/4885HPGD 1157/4885ALDH1A1 298/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.