SCHEMBL11225822

SCHEMBL11225822

COc1cc2c(cc1OC)C(C(C)CCCl)OCC2

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC18A2 Q05940 3/20 0.40
KCNN2 Q9H2S1 4/20 0.39
KCNN3 Q9UGI6 4/20 0.39
KCNN1 Q92952 2/20 0.39
KDM4E B2RXH2 3/20 0.39
ALDH1A1 P00352 3/20 0.39
HSD17B10 Q99714 3/20 0.39
LMNA P02545 2/20 0.39
MAPK1 P28482 2/20 0.39
CYP2D6 P10635 1/20 0.39
MAOA P21397 2/20 0.39
TSHR P16473 2/20 0.38
ABCB11 O95342 1/20 0.37
POLB P06746 1/20 0.37
HTR1A P08908 1/20 0.37
ADRA2A P08913 1/20 0.37
MAPT P10636 1/20 0.37
HPGD P15428 1/20 0.37
SCN1A P35498 1/20 0.37
HTR2B P41595 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11221051 0.92 SLC18A2 (0.39) SLC18A2KCNN2KCNN3KCNN1KDM4E
SCHEMBL11225508 0.80 KCNN2 (0.39) SLC18A2KCNN2KCNN3KCNN1KDM4E
SCHEMBL11221677 0.77 SLC18A2 (0.39) SLC18A2KCNN2KCNN3KCNN1KDM4E
SCHEMBL9688216 0.75 KCNN2 (0.43) KCNN2KCNN3KCNN1KDM4EALDH1A1
SCHEMBL7290833 0.75 ALDH1A1 (0.43) KCNN2KCNN3KCNN1KDM4EALDH1A1
SCHEMBL11370360 0.74 MAOA (0.41) SLC18A2KCNN2KCNN3KCNN1MAOA
SCHEMBL11220353 0.74 MAOA (0.41) SLC18A2KCNN2KCNN3KCNN1MAOA
SCHEMBL11224266 0.74 SLC18A2 (0.38) SLC18A2KCNN2KCNN3KCNN1KDM4E
SCHEMBL11222256 0.73 KCNN2 (0.38) SLC18A2KCNN2KCNN3KCNN1KDM4E
SCHEMBL11220460 0.73 KCNN2 (0.44) KCNN2KCNN3KCNN1ALDH1A1MAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4352805-A BENZOXEPINE DERIVATIVES THE UPJOHN COMPANY (US) 1982-10-05 US disclosed
US-4312868-A HYPOTENSIVE, ANTIPSYCHOTIC THE UPJOHN COMPANY (US) 1982-01-26 US disclosed
US-4251526-A HYPOTENSIVE AGENTS AND ANTIPSYCHOTIC PHARMACIA & UPJOHN COMPANY 1981-02-17 US disclosed
US-4250175-A HYPOTENSIVE AGENTS, ANTIDEPRESSANTS PHARMACIA & UPJOHN COMPANY 1981-02-10 US disclosed
US-4250181-A HYPOTENSIVE AGENTS, ANTIDEPRESSANTS THE UPJOHN COMPANY (US) 1981-02-10 US disclosed
US-4247553-A HYPOTENSIVE AGENTS, ANTIDEPRESSANTS THE UPJOHN COMPANY (US) 1981-01-27 US disclosed
US-4181665-A INTERMEDIATES FOR AMINO DERIVATIVES POSSESSING HYPOTENSIVE AND CENTRAL NERVOUS SYSTEM ACTIVITY THE UPJOHN COMPANY (US) 1980-01-01 US disclosed
US-4179510-A ISOCHROMANS AND 2-BENZOXEPINS THE UPJOHN COMPANY (US) 1979-12-18 US disclosed
US-4153612-A 2-Benzoxepins THE UPJOHN COMPANY (US) 1979-05-08 US disclosed