SCHEMBL11225918

SCHEMBL11225918

C#Cc1ccc(CC(C)C)c([N+](=O)[O-])c1

nearest known ligand 0.55

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
FBP1 P09467 4/20 0.43
ALOX15 P16050 1/20 0.42
ALOX12 P18054 1/20 0.42
PDK1 Q15118 1/20 0.38
VCAM1 P19320 2/20 0.36
CYP1A2 P05177 1/20 0.35
P2RY6 Q15077 1/20 0.33
SNCA P37840 1/20 0.33
CYP2C9 P11712 1/20 0.33
MAPT P10636 2/20 0.32
ALDH1A1 P00352 1/20 0.32
HTT P42858 1/20 0.32
POLB P06746 1/20 0.32
CYP2C19 P33261 1/20 0.32
MAPK1 P28482 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11702124 0.83 ALOX15 (0.36) FBP1ALOX15ALOX12PDK1VCAM1
SCHEMBL3032856 0.78 CYP1A2 (0.57) FBP1ALOX15ALOX12CYP1A2MAPT
SCHEMBL10019205 0.78 TSHR (0.56) FBP1ALOX15ALOX12PDK1CYP1A2
SCHEMBL11807538 0.78 GABRA1 (0.47) FBP1ALOX15ALOX12PDK1CYP1A2
SCHEMBL2064927 0.76 FBP1 (0.46) FBP1ALOX15ALOX12PDK1CYP1A2
SCHEMBL10019199 0.76 TDP1 (0.49) FBP1ALOX15ALOX12PDK1CYP1A2
SCHEMBL11229564 0.76 PDK1 (0.50) ALOX15ALOX12PDK1VCAM1P2RY6
SCHEMBL11689602 0.75 TSHR (0.50) VCAM1CYP1A2P2RY6CYP2C9MAPT
SCHEMBL13269178 0.74 ALDH5A1 (0.53) FBP1ALOX15ALOX12PDK1VCAM1
SCHEMBL10019202 0.73 MAPK1 (0.52) ALOX15MAPTALDH1A1POLBMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 22 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4150148-A NITROSUBSTITUTED WILLIAM H. RORER, INC. (US) 1979-04-17 US claimed
US-3981932-A Ethynylbenzene compounds and derivatives thereof WILLIAM H. RORER, INC. (US) 1976-09-21 US claimed
US-4365093-A Ethynylbenzene compounds and derivatives thereof WILLIAM H. RORER, INC. (US) 1982-12-21 US disclosed
US-4296264-A Ethynylbenzene compounds and derivatives thereof WILLIAM H. RORER, INC. (US) 1981-10-20 US disclosed
US-4288457-A Ethynylbenzene compounds and derivatives thereof WILLIAM H. RORER, INC. (US) 1981-09-08 US disclosed
US-4264627-A Ethynylbenzene compounds and derivatives thereof to treat inflammation, pain or fever WILLIAM H. RORER, INC. (US) 1981-04-28 US disclosed
US-4171373-A Ethynylbenzene compounds and derivatives thereof to treat pain, fever and inflammation WILLIAM H. RORER, INC. (US) 1979-10-16 US disclosed
US-4168320-A Ethynylbenzene compounds and derivatives thereof to treat inflammation, pain or fever WILLIAM H. RORER, INC. (US) 1979-09-18 US disclosed
US-4166133-A ETHYNYLBENZENE COMPOUNDS AND DERIVATIVES THEREOF TO TREAT PAIN, FEVER AND INFLAMMATION WILLIAM H. RORER, INC. (US) 1979-08-28 US disclosed
US-4157449-A Ethynylbenzene compounds and derivatives thereof WILLIAM H. RORER, INC. (US) 1979-06-05 US disclosed
US-4150148-A NITROSUBSTITUTED WILLIAM H. RORER, INC. (US) 1979-04-17 US disclosed
US-4105786-A ANTIINFLAMMATORY WILLIAM H. RORER, INC. (US) 1978-08-08 US disclosed
US-4101591-A Ethynylbenzene compounds and derivatives thereof WILLIAM H. RORER, INC. (US) 1978-07-18 US disclosed
US-4096279-A Ethynylbenzene compounds and derivatives thereof in the treatment of pain fever and inflammation WILLIAM H. RORER, INC. (US) 1978-06-20 US disclosed
US-4094995-A ETHYNYLBENZENE COMPOUNDS AND DERIVATIVES THEREOF TO TREAT PAIN, FEVER AND INFLAMMATION WILLIAM H. RORER, INC. (US) 1978-06-13 US disclosed
US-4093737-A Ethynylbenzene compounds and derivatives thereof in the treatment of pain, fever or inflammation WILLIAM H. RORER, INC. (US) 1978-06-06 US disclosed
US-4075354-A ETHYNYLBENZENE COMPOUNDS AND DERIVATIVES THEREOF FOR TREATING PAIN FEVER AND INFLAMMATION WILLIAM H. RORER, INC. (US) 1978-02-21 US disclosed
US-4016214-A Preparation of ethynylbenzenes WILLIAM H. RORER, INC. (US) 1977-04-05 US disclosed
US-3981932-A Ethynylbenzene compounds and derivatives thereof WILLIAM H. RORER, INC. (US) 1976-09-21 US disclosed
US-3952067-A Ethynylbenzenes WILLIAM H. RORER, INC. (US) 1976-04-20 US disclosed