SCHEMBL11228381

SCHEMBL11228381

Cc1cc2c(cc1C)OC(CCBr)CO2

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 1/20 0.40
CA2 P00918 4/20 0.38
HTT P42858 1/20 0.37
MAPT P10636 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.35
IMPDH2 P12268 1/20 0.35
IMPDH1 P20839 1/20 0.35
GAA P10253 1/20 0.34
HSD17B10 Q99714 1/20 0.34
HTR6 P50406 1/20 0.33
POLB P06746 1/20 0.33
ESR2 Q92731 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11235851 0.83 CA2 (0.56) MTNR1ACA2HTTMAPTTDP1
SCHEMBL11222928 0.83 CA2 (0.49) CA2HTTMAPTTDP1GAA
SCHEMBL11224196 0.77 CA2 (0.56) MTNR1ACA2HTTMAPTSMN1; SMN2
SCHEMBL11230966 0.77 CA2 (0.56) CA2HTTMAPTSMN1; SMN2
SCHEMBL11232203 0.77 MTNR1A (0.57) MTNR1AMAPTTDP1GAAPOLB
SCHEMBL11219443 0.77 MTNR1A (0.64) MTNR1AMAPTTDP1GAAPOLB
SCHEMBL5871673 0.76 HTT (0.61) MTNR1ACA2HTTSMN1; SMN2POLB
SCHEMBL17272101 0.75 HTT (0.37) CA2HTTSMN1; SMN2POLB
SCHEMBL11026135 0.69 CA2 (0.55) CA2
SCHEMBL17272701 0.69 CA2 (0.58) CA2MAPTGAAHTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4353901-A HYPERTENSION, CONGESTIVE HEART FAILURE, ARRHYTHMIAMIGRAINE, VASOSPASTIC DISORDERS, ASTHMA SYNTEX (U.S.A.) INC. (US) 1982-10-12 US disclosed