SCHEMBL11229323

SCHEMBL11229323

CCc1nc(Cl)c(C#N)cc1-c1ccnc(C)c1

nearest known ligand 0.46

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
MTOR P42345 3/20 0.41
WNT3A P56704 3/20 0.40
LRRK2 Q5S007 3/20 0.40
ALDH1A1 P00352 1/20 0.39
AAK1 Q2M2I8 2/20 0.38
CYP3A4 P08684 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11236432 0.84 PDE3B (0.51) CYP1A2CYP2C9CYP2C19NPSR1ALDH1A1
SCHEMBL11241191 0.82 WNT3A (0.45) MTORWNT3ALRRK2AAK1CYP3A4
SCHEMBL7273135 0.82 MTOR (0.42) MTORAAK1
SCHEMBL11230737 0.80 MTOR (0.40) MTORAAK1
SCHEMBL11226168 0.77 ALDH1A1 (0.49) CYP1A2CYP2C9CYP2C19NPSR1ALDH1A1
SCHEMBL11396219 0.76 FTO (0.44) MTORWNT3A
SCHEMBL7270939 0.75 MTOR (0.45) MTOR
SCHEMBL11236490 0.75 NCOA1 (0.39) NPSR1MTORALDH1A1CYP3A4
SCHEMBL11166411 0.75 PIK3CB (0.47) MTORAAK1
SCHEMBL11241603 0.74 PDE3B (0.53) CYP1A2CYP2C9CYP2C19NPSR1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4361568-A 5-(Pyridinyl)-1H-pyrazolo[3,4-b]pyridin-3-amines and their cardiotonic use STERLING DRUG INC. (US) 1982-11-30 US disclosed
US-4264603-A 5-(Pyridinyl)-1H-pyrazolo[3,4-b]pyridine-3-amines, their use as cardiotonics and their preparation STERLING DRUG INC. (US) 1981-04-28 US disclosed