SCHEMBL11235100

SCHEMBL11235100

COc1ccc2c(c1)OC(C(O)CN1CCC3(CC1)CNC(=O)CO3)CO2

nearest known ligand 0.49

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 2/20 0.38
HTR2A P28223 1/20 0.37
LMNA P02545 1/20 0.35
LRRK2 Q5S007 2/20 0.35
FFAR1 O14842 1/20 0.35
CCR1 P32246 3/20 0.35
DRD2 P14416 2/20 0.35
DRD4 P21917 2/20 0.35
KCNH2 Q12809 1/20 0.34
HTR1A P08908 1/20 0.34
HTR7 P34969 1/20 0.34
SIGMAR1 Q99720 1/20 0.33
CYP3A4 P08684 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11224382 0.97 HTR2A (0.37) MTNR1AHTR2ALMNALRRK2CCR1
SCHEMBL11231912 0.89 CCR1 (0.34) CCR1DRD2DRD4KCNH2
SCHEMBL11224230 0.87 CCR1 (0.42) CCR1KCNH2
SCHEMBL11224028 0.86 CCR1 (0.32) LRRK2CCR1DRD2KCNH2
SCHEMBL11220558 0.86 DRD2 (0.40) HTR2ALMNACCR1DRD2DRD4
SCHEMBL11227376 0.85 CCR1 (0.34) LRRK2CCR1DRD2DRD4KCNH2
SCHEMBL11223663 0.83 CCR1 (0.42) CCR1KCNH2
SCHEMBL11221152 0.82 MTNR1A (0.48) MTNR1AHTR2ALRRK2FFAR1DRD2
SCHEMBL11230978 0.78 MTNR1A (0.44) MTNR1AHTR2ALRRK2FFAR1DRD2
SCHEMBL10992228 0.75 SLC6A2 (0.40) MTNR1ALMNAFFAR1SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4353901-A HYPERTENSION, CONGESTIVE HEART FAILURE, ARRHYTHMIAMIGRAINE, VASOSPASTIC DISORDERS, ASTHMA SYNTEX (U.S.A.) INC. (US) 1982-10-12 US disclosed