SCHEMBL11235309

SCHEMBL11235309

CCOC(=O)c1cc(-c2cc(C)cc(C)n2)c(C)[nH]c1=O

nearest known ligand 0.58

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.58
L3MBTL1 Q9Y468 3/20 0.58
MAPT P10636 3/20 0.58
LMNA P02545 2/20 0.58
POLB P06746 3/20 0.51
GAA P10253 2/20 0.51
NPC1 O15118 1/20 0.51
CDK5 Q00535 5/20 0.47
CDK5R1 Q15078 5/20 0.47
KDM4E B2RXH2 5/20 0.45
TDP1 Q9NUW8 1/20 0.45
KMT2A Q03164 1/20 0.44
PDE3B Q13370 1/20 0.40
PDE3A Q14432 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11233196 0.83 KDM4E (0.51) ALDH1A1L3MBTL1MAPTLMNAPOLB
SCHEMBL11238700 0.82 POLB (0.39) ALDH1A1L3MBTL1MAPTLMNAPOLB
SCHEMBL9671945 0.75 ALDH1A1 (1.00) ALDH1A1L3MBTL1MAPTLMNAPOLB
SCHEMBL11242636 0.74 CDK5 (0.62) ALDH1A1L3MBTL1MAPTLMNAPOLB
SCHEMBL11231843 0.73 PDE3B (0.51) LMNAGAANPC1KDM4EKMT2A
SCHEMBL11243686 0.73 KDM4E (0.36) ALDH1A1MAPTLMNAPOLBKDM4E
SCHEMBL31555544 0.72 KMT2A (0.41) ALDH1A1MAPTLMNAPOLBGAA
SCHEMBL9476375 0.71 GAA (0.88) ALDH1A1L3MBTL1MAPTLMNAPOLB
SCHEMBL10004177 0.71 ALDH1A1 (0.73) ALDH1A1L3MBTL1MAPTLMNAPOLB
SCHEMBL9672980 0.70 ALDH1A1 (0.88) ALDH1A1L3MBTL1MAPTLMNAPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4312875-A 5-(Pyridinyl)-6-(lower-alkyl)-2(1H)-pyridinones, 1,2-dihydro-2-oxo-5-(pyridinyl)-6-(lower-alkyl)nicotinic acids and lower-alkyl esters thereof, and cardiotonic use thereof STERLING DRUG INC. (US) 1982-01-26 US disclosed