SCHEMBL11243686

SCHEMBL11243686

Cc1cc(C)nc(-c2cc(Cl)c(=O)[nH]c2C)c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.36
RXFP1 Q9HBX9 1/20 0.36
GRIN2D O15399 2/20 0.35
GRIN3B O60391 2/20 0.35
GRIN1 Q05586 2/20 0.35
GRIN2A Q12879 2/20 0.35
GRIN2B Q13224 2/20 0.35
GRIN2C Q14957 2/20 0.35
GRIN3A Q8TCU5 2/20 0.35
IDH1 O75874 1/20 0.34
TP53 P04637 2/20 0.33
POLB P06746 2/20 0.33
SMN1; SMN2 Q16637 3/20 0.33
HTT P42858 2/20 0.33
MAPK1 P28482 1/20 0.33
KMT2A Q03164 3/20 0.32
MEN1 O00255 2/20 0.32
LMNA P02545 2/20 0.32
HPGD P15428 2/20 0.32
HSD17B10 Q99714 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11231843 0.81 PDE3B (0.51) KDM4ERXFP1KMT2AMEN1LMNA
SCHEMBL11233196 0.78 KDM4E (0.51) KDM4ERXFP1POLBSMN1; SMN2MAPK1
SCHEMBL11232009 0.78 KDM4E (0.61) KDM4ERXFP1KMT2AMEN1LMNA
SCHEMBL11238700 0.77 POLB (0.39) KDM4ERXFP1POLBKMT2AMEN1
SCHEMBL11240531 0.74 CA12 (0.39) KDM4ETP53SMN1; SMN2HTTMAPK1
SCHEMBL11235309 0.73 ALDH1A1 (0.58) KDM4EPOLBKMT2ALMNAALDH1A1
SCHEMBL11235848 0.68 PDE3B (0.67) KDM4ELMNAHPGDALDH1A1MAPT
SCHEMBL1426158 0.67 GRIN2D (0.45) KDM4EGRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL29648194 0.66 NOS3 (0.55) KDM4EPOLBSMN1; SMN2KMT2AMEN1
SCHEMBL3084862 0.66 NOS3 (0.55) KDM4EPOLBSMN1; SMN2KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4365065-A 1-(Pyridinyl)-2-(dimethylamino)ethenyl lower-alkyl ketones STERLING DRUG INC. (US) 1982-12-21 US disclosed
US-4313951-A 3-Substituted-6-(lower-alkyl)-5-(pyridinyl)-2(1H)-pyridinones, their cardiotonic use and intermediates therefor STERLING DRUG INC. (US) 1982-02-02 US disclosed