SCHEMBL11240004

SCHEMBL11240004

CC(C)Cc1ccc2sc3cc(CC(=O)O)ccc3c2c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.44
HPGD P15428 5/20 0.44
HSD17B10 Q99714 5/20 0.44
ALDH1A1 P00352 4/20 0.44
MAPT P10636 3/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
TSHR P16473 3/20 0.40
PFKFB3 Q16875 1/20 0.38
PTGS1 P23219 4/20 0.38
PTGS2 P35354 3/20 0.38
LMNA P02545 3/20 0.38
AKR1C3 P42330 3/20 0.38
CYP2C9 P11712 2/20 0.38
CXCR1 P25024 2/20 0.38
CXCR2 P25025 2/20 0.38
NFKB1 P19838 2/20 0.38
BLM P54132 2/20 0.38
PMP22 Q01453 2/20 0.38
AKR1C2 P52895 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11237206 0.85 KDM4E (0.47) KDM4EHPGDHSD17B10ALDH1A1MAPT
SCHEMBL11248260 0.84 NPC1 (0.46) MAPTNFKB1GABRA1GABRB2
SCHEMBL11243330 0.83 SLC22A12 (0.45) KDM4EHPGDHSD17B10ALDH1A1MAPT
SCHEMBL24476988 0.81 GABRA1 (0.46) KDM4EHPGDHSD17B10ALDH1A1MAPT
SCHEMBL11246646 0.80 CA2 (0.49) KDM4EHPGDHSD17B10ALDH1A1MAPT
SCHEMBL26082534 0.80 GABRA1 (0.38) KDM4EHPGDALDH1A1MAPTMEN1
SCHEMBL11253323 0.80 CYP1A2 (0.47) KDM4EHPGDHSD17B10ALDH1A1MAPT
SCHEMBL11240017 0.79 KEAP1 (0.51) KDM4EHPGDHSD17B10ALDH1A1MAPT
SCHEMBL11246422 0.79 KDM4E (0.44) KDM4EHPGDHSD17B10ALDH1A1MAPT
SCHEMBL11244551 0.79 KDM4E (0.44) KDM4EHPGDHSD17B10ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4334078-A ANTIINFLAMMATORY AGENTS, ANALGESICS, ANTIRHEUMATICS HOFFMANN-LA ROCHE INC. (US) 1982-06-08 US disclosed
US-4219657-A USED AS ANTIINFLAMATORY AGENTS, ANALGESICS, ANTIRHEUMATIC AGENTS HOFFMANN-LA ROCHE INC. (US) 1980-08-26 US disclosed