SCHEMBL11241295

SCHEMBL11241295

CC(=O)N1CCC(OC(=O)O)(c2ccccc2Oc2ccc(F)cc2)CC1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
USP2 O75604 2/20 0.40
ALDH1A1 P00352 4/20 0.39
CYP2C19 P33261 3/20 0.39
MAPK1 P28482 2/20 0.39
MMP2 P08253 2/20 0.39
MMP9 P14780 2/20 0.39
KCNA3 P22001 1/20 0.39
CYP2D6 P10635 4/20 0.38
TSHR P16473 1/20 0.38
MEN1 O00255 1/20 0.38
RAB9A P51151 1/20 0.38
KMT2A Q03164 1/20 0.38
GAA P10253 1/20 0.38
GFER P55789 1/20 0.38
CYP3A4 P08684 3/20 0.38
CYP2C9 P11712 2/20 0.38
CYP1A2 P05177 1/20 0.37
HPGD P15428 1/20 0.37
ALOX12 P18054 1/20 0.37
HSD17B10 Q99714 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11243000 0.93 USP2 (0.43) USP2ALDH1A1CYP2C19MAPK1MMP2
SCHEMBL11255005 0.88 SCN1A (0.41) ALDH1A1HPGDHTR1ASLC6A2SLC6A4
SCHEMBL11241289 0.84 KMT2A (0.44) USP2ALDH1A1CYP2C19MAPK1MMP2
SCHEMBL11239682 0.81 SLC6A2 (0.44) ALDH1A1MAPK1HTR1ASLC6A2SLC6A4
Bromide SCHEMBL11242341 0.80 SLC6A2 (0.43) ALDH1A1MAPK1HTR1ASLC6A2SLC6A4
SCHEMBL11248847 0.80 ITGAL (0.41) USP2ALDH1A1CYP2C19MAPK1KCNA3
SCHEMBL11246085 0.78 MMP1 (0.43) ALDH1A1MMP9MEN1KMT2AHPGD
SCHEMBL11471965 0.76 MEN1 (0.43) USP2ALDH1A1CYP2C19MAPK1MMP2
SCHEMBL11242994 0.76 USP2 (0.45) USP2ALDH1A1CYP2C19MAPK1MMP2
SCHEMBL11486442 0.76 USP2 (0.45) USP2ALDH1A1CYP2C19MAPK1MMP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0016261-B1 SPIRO(DIBENZ(B,F)OXEPIN-PIPERIDINES) AND METHODS OF PREPARING SAME HOECHST AKTIENGESELLSCHAFT (DE) 1982-12-29 EP disclosed
EP-0016261-A1 Spiro(dibenz(b,f)oxepin-piperidines) and methods of preparing same HOECHST AKTIENGESELLSCHAFT (DE) 1980-10-01 EP disclosed