SCHEMBL11242343

SCHEMBL11242343

CNC(N)=NC(=O)C(Br)c1c(Cl)cccc1Cl

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 2/20 0.36
KMT2A Q03164 2/20 0.36
LMNA P02545 2/20 0.36
CYP2D6 P10635 2/20 0.36
HIF1A Q16665 2/20 0.36
MEN1 O00255 1/20 0.36
CYP3A4 P08684 1/20 0.36
HTR1A P08908 1/20 0.36
CYP2C9 P11712 1/20 0.36
ADRA2B P18089 1/20 0.36
ADRA2C P18825 1/20 0.36
MAOA P21397 1/20 0.36
ADRA1D P25100 1/20 0.36
HTR2A P28223 1/20 0.36
HTR2C P28335 1/20 0.36
MAPK1 P28482 1/20 0.36
CYP2C19 P33261 1/20 0.36
ADRA1A P35348 1/20 0.36
DRD3 P35462 1/20 0.36
OPRK1 P41145 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11249700 0.83 HTR2B (0.47) ADRA2AKMT2ALMNACYP2D6HIF1A
SCHEMBL11246671 0.79 ADRA2A (0.36) ADRA2AKMT2ALMNACYP2D6HIF1A
SCHEMBL11247965 0.79 NPC1 (0.38) ADRA2AKMT2ALMNACYP2D6HIF1A
SCHEMBL11239762 0.79 ADRA2A (0.36) ADRA2AKMT2ALMNACYP2D6HIF1A
SCHEMBL5179498 0.70 ALDH1A1 (0.40) KMT2ALMNACYP2D6HIF1ABLM
SCHEMBL11244852 0.70 POLB (0.34) KMT2AMEN1MAPK1POLBALDH1A1
SCHEMBL11263022 0.70 POLB (0.34) KMT2AMEN1MAPK1POLBALDH1A1
SCHEMBL9125705 0.69 KMT2A (0.40) KMT2ACYP2D6HIF1AMEN1CYP3A4
SCHEMBL11241971 0.68 ALDH1A1 (0.41) KMT2AMEN1POLBALDH1A1CYP1A2
SCHEMBL11247894 0.68 TSHR (0.42) KMT2AMEN1ALDH1A1CXCL8TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4318915-A Substituted guandines and methods of preparation thereof BEIERSDORF AKTIENGESELLSCHAFT (DE) 1982-03-09 US claimed
US-4318915-A Substituted guandines and methods of preparation thereof BEIERSDORF AKTIENGESELLSCHAFT (DE) 1982-03-09 US disclosed