SCHEMBL11249700

SCHEMBL11249700

NC(N)=NC(=O)C(Br)c1c(Cl)cccc1Cl

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2B P41595 4/20 0.47
ADRA2A P08913 3/20 0.47
LMNA P02545 2/20 0.47
CYP2D6 P10635 2/20 0.47
HIF1A Q16665 2/20 0.47
HTR1A P08908 2/20 0.47
ADRA2B P18089 2/20 0.47
ADRA2C P18825 2/20 0.47
MAOA P21397 2/20 0.47
ADRA1D P25100 2/20 0.47
HTR2A P28223 2/20 0.47
HTR2C P28335 2/20 0.47
ADRA1A P35348 2/20 0.47
DRD3 P35462 2/20 0.47
NISCH Q9Y2I1 2/20 0.47
MEN1 O00255 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2C9 P11712 1/20 0.47
MAPK1 P28482 1/20 0.47
CYP2C19 P33261 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11239762 0.83 ADRA2A (0.36) HTR2BADRA2ALMNACYP2D6HIF1A
SCHEMBL11246671 0.83 ADRA2A (0.36) HTR2BADRA2ALMNACYP2D6HIF1A
SCHEMBL11247965 0.83 NPC1 (0.38) HTR2BADRA2ALMNACYP2D6HIF1A
SCHEMBL11242343 0.83 ADRA2A (0.36) HTR2BADRA2ALMNACYP2D6HIF1A
SCHEMBL11249016 0.81 ADRA2A (0.49) HTR2BADRA2ALMNACYP2D6HIF1A
Hydrochloric Acid SCHEMBL11256890 0.74 ADRA2A (0.45) HTR2BADRA2ALMNACYP2D6HIF1A
SCHEMBL11241971 0.74 ALDH1A1 (0.41) MEN1KMT2APOLBCYP1A2TSHR
SCHEMBL11247894 0.74 TSHR (0.42) MEN1KMT2ATSHR
SCHEMBL5179498 0.72 ALDH1A1 (0.40) LMNACYP2D6HIF1AKMT2ABLM
SCHEMBL11245746 0.71 CYP3A4 (0.31) CYP3A4CYP2C19MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4318915-A Substituted guandines and methods of preparation thereof BEIERSDORF AKTIENGESELLSCHAFT (DE) 1982-03-09 US disclosed