SCHEMBL1124372

SCHEMBL1124372

O=Cc1ccc(N2CCOCC2)nc1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.55
HPGD P15428 3/20 0.55
CYP1A2 P05177 1/20 0.55
CYP2C9 P11712 1/20 0.55
HSD17B10 Q99714 3/20 0.51
KDM4E B2RXH2 2/20 0.51
SMN1; SMN2 Q16637 2/20 0.51
MAPT P10636 2/20 0.51
MEN1 O00255 1/20 0.51
LMNA P02545 1/20 0.51
GAA P10253 1/20 0.51
HTT P42858 1/20 0.51
RECQL P46063 1/20 0.51
KMT2A Q03164 1/20 0.51
TDP1 Q9NUW8 1/20 0.51
ALDH3A1 P30838 1/20 0.50
ALDH1A3 P47895 1/20 0.50
POLB P06746 1/20 0.50
ALOX15 P16050 1/20 0.50
ERN1 O75460 2/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30287647 1.00 ALDH1A1 (0.55) ALDH1A1HPGDCYP1A2CYP2C9HSD17B10
SCHEMBL1735017 0.84 TRIM24 (0.53) ALDH1A1KDM4ESMN1; SMN2MAPTLMNA
SCHEMBL4768589 0.83 ALDH1A1 (0.51) ALDH1A1HPGDCYP1A2CYP2C9HSD17B10
SCHEMBL840830 0.83 ALDH1A1 (0.55) ALDH1A1KDM4ESMN1; SMN2MAPTLMNA
SCHEMBL4647849 0.81 ALDH1A1 (0.55) ALDH1A1HPGDCYP1A2CYP2C9HSD17B10
SCHEMBL25082375 0.80 KCNJ1 (0.41) ALDH1A1HPGDCYP1A2CYP2C9HSD17B10
SCHEMBL29805413 0.80 PLD1 (0.49) ALDH1A1CYP1A2HSD17B10KDM4EHTT
SCHEMBL1569943 0.80 PLD1 (0.49) ALDH1A1CYP1A2HSD17B10KDM4EHTT
SCHEMBL2322917 0.80 ALDH1A1 (0.57) ALDH1A1SMN1; SMN2MAPTKMT2ATDP1
SCHEMBL3786488 0.79 PIM2 (0.54) ALDH1A1HPGDCYP1A2CYP2C9HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 190 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10787484-B2 Compositions and methods for treating cardiovascular disease GENENTECH, INC. (US) 2020-09-29 US claimed
US-20190177366-A1 COMPOSITIONS AND METHODS FOR TREATING CARDIOVASCULAR DISEASE GENENTECH, INC. (US) 2019-06-13 US claimed
US-20260103444-A1 8-HYDROXYQUINOLINE COMPOUND AND USE THEREOF UNIV OSAKA (JP) 2026-04-16 US disclosed
EP-4599832-A1 8-HYDROXYQUINOLINE COMPOUND AND USE THEREOF OSAKA UNIVERSITY (JP) 2025-08-13 EP disclosed
EP-3759075-B1 COMPOUNDS WITH FERROPTOSIS INDUCING ACTIVITY AND METHODS OF THEIR USE FERRO THERAPEUTICS INC (US) 2025-07-23 EP disclosed
CN-119968204-A 8-Hydroxyquinoline compound and use thereof 国立大学法人大阪大学 2025-05-09 CN disclosed
US-20250114374-A1 BCL-2 INHIBITORS NEWAVE PHARMACEUTICAL INC. 2025-04-10 US disclosed
US-20250099481-A1 BCL-2 INHIBITORS NEWAVE PHARMACEUTICAL INC. 2025-03-27 US disclosed
WO-2024075815-A1 8-HYDROXYQUINOLINE COMPOUND AND USE THEREOF 国立大学法人大阪大学 2024-04-11 WO disclosed
CN-114828959-B 3- (5-methoxy-1-oxo-isoindolin-2-yl) piperidine-2, 6-dione derivative and application thereof 诺华股份有限公司 2024-04-02 CN disclosed
EP-4076650-B1 3-(5-METHOXY-1-OXOISOINDOLIN-2-YL)PIPERIDINE-2,6-DIONE DERIVATIVES AND USES THEREOF NOVARTIS AG (CH) 2024-02-28 EP disclosed
US-20080242597-A1 Antibiotic compounds MERCK SHARP & DOHME CORP. 2008-10-02 US disclosed
US-20080242597-A1 Antibiotic compounds MERCK SHARP & DOHME CORP. 2008-10-02 US disclosed
US-20080242597-A1 Antibiotic compounds MERCK SHARP & DOHME CORP. 2008-10-02 US disclosed
US-20080176883-A1 Antiinflammtory, antiproliferative, anticancer agents; (3-Hydroxy-pyrrolidin-1-yl)-(3-trifluoromethyl-7,8-dihydro-5H-[1,6]naphthyridin-6-yl)-methanone ABBVIE INC. 2008-07-24 US disclosed
WO-2008035049-A1 ADAMANTANYL-(CYCLOPROPYL)-KETONES AS METABOTROPIC GLUTAMATE RECEPTOR MODULATORS MERZ PHARMA GMBH & CO. KGAA (DE) 2008-03-27 WO disclosed
US-20080039452-A1 Fused Quinoline Derivative and Use Thereof TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-02-14 US disclosed
WO-2007134958-A1 THIAZOLO-PYRAMIDINE / PYRIDINE UREA DERIVATIVES AS ADENOSINE A2B RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2007-11-29 WO disclosed
US-20070270433-A1 Thiazolo-pyrimidine/pyridine urea derivatives BRINKMAN JOHN A 2007-11-22 US disclosed
WO-2007073935-A1 HETEROCYCLIC COMPOUNDS LEK PHARMACEUTICALS D.D. (SI) 2007-07-05 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (9 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080176883-A1 Antiinflammtory, antiproliferative, anticancer agents; (3-Hydroxy-pyrrolidin-1-yl)-(3-trifluoromethyl-7,8-dihydro-5H-[1,6]naphthyridin-6-yl)-methanone MIF, CCL5, CCR2 ALDH1A1 433/4885HPGD 65/4885CYP1A2 834/4885
US-20250114374-A1 BCL-2 INHIBITORS BCL2, BCL2L1, BCL2L10 ALDH1A1 3831/4885HPGD 3983/4885CYP1A2 2936/4885
US-20250099481-A1 BCL-2 INHIBITORS BCL2, BCL2L1, BCL2L10 ALDH1A1 3478/4885HPGD 3819/4885CYP1A2 2579/4885
US-20260103444-A1 8-HYDROXYQUINOLINE COMPOUND AND USE THEREOF MYLK2, MYLK, ATP2A1 ALDH1A1 2735/4885HPGD 1407/4885CYP1A2 1775/4885
US-20070270433-A1 Thiazolo-pyrimidine/pyridine urea derivatives ADORA2B, UTS2R, TBXA2R ALDH1A1 676/4885HPGD 1175/4885CYP1A2 1385/4885
US-20080039452-A1 Fused Quinoline Derivative and Use Thereof TACR2, HRH3, HRH2 ALDH1A1 2917/4885HPGD 1619/4885CYP1A2 1194/4885
US-10787484-B2 Compositions and methods for treating cardiovascular disease PCSK9, PCSK7, PCSK6 ALDH1A1 4023/4885HPGD 2382/4885CYP1A2 3180/4885
US-20190177366-A1 COMPOSITIONS AND METHODS FOR TREATING CARDIOVASCULAR DISEASE PCSK9, PCSK7, PCSK6 ALDH1A1 4023/4885HPGD 2382/4885CYP1A2 3180/4885
US-20080242597-A1 Antibiotic compounds PEPD, NRDC, MRPL21 ALDH1A1 4047/4885HPGD 3228/4885CYP1A2 4229/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.